SCHEMBL4457030

SCHEMBL4457030

c1ccc(-c2cccc3[nH]c(-c4cccc(-c5nc6c(-c7ccccc7)cccc6[nH]5)c4)nc23)cc1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 5/20 0.53
PARP1 P09874 6/20 0.51
GAA P10253 5/20 0.51
MGAM O43451 4/20 0.51
SI P14410 4/20 0.51
MGAM2 Q2M2H8 4/20 0.51
NPC1 O15118 3/20 0.49
RAB9A P51151 3/20 0.49
PDE10A Q9Y233 1/20 0.48
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 2/20 0.47
HPGD P15428 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
TP53 P04637 1/20 0.47
HSD17B10 Q99714 1/20 0.47
CNR2 P34972 1/20 0.47
VSIR Q9H7M9 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL230979 0.97 DHODH (0.53) DHODHPARP1GAAMGAMSI
SCHEMBL31027957 0.93 DHODH (0.59) DHODHPARP1GAAMGAMSI
SCHEMBL9346643 0.93 GAA (0.54) DHODHPARP1GAAMGAMSI
SCHEMBL7146754 0.91 DHODH (0.62) DHODHPARP1GAAMGAMSI
SCHEMBL1170898 0.91 DHODH (0.54) DHODHPARP1GAAMGAMSI
SCHEMBL8818524 0.89 MGAM (0.68) DHODHPARP1GAAMGAMSI
SCHEMBL8817536 0.89 NR1I3 (0.58) DHODHPARP1GAAMGAMSI
SCHEMBL8816555 0.89 DHODH (0.51) DHODHPARP1GAAMGAMSI
SCHEMBL8891044 0.89 MGAM (0.68) DHODHPARP1GAAMGAMSI
SCHEMBL8816885 0.87 DHODH (0.50) DHODHPARP1GAAMGAMSI

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125752-A1 HETEROCYCLIC BRIDGED BIPHENYLS BASF SE (DE) 2009-12-02 EP disclosed
WO-2008119666-A1 HETEROCYCLIC BRIDGED BIPHENYLS BASF SE (CH) 2008-10-09 WO disclosed