SCHEMBL4457039

SCHEMBL4457039

Cc1cc2c(cc1Br)OC(c1ccccc1)(c1ccccc1)O2

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 11/20 0.47
ALDH1A1 P00352 1/20 0.34
NPSR1 Q6W5P4 3/20 0.33
CYP1A2 P05177 3/20 0.32
CYP3A4 P08684 3/20 0.32
CYP2C9 P11712 3/20 0.32
CYP2C19 P33261 3/20 0.32
CYP2D6 P10635 1/20 0.32
HTT P42858 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
HSP90AA1 P07900 1/20 0.31
SIRT1 Q96EB6 1/20 0.30
MAP3K14 Q99558 1/20 0.30
SRD5A1 P18405 1/20 0.30
SRD5A2 P31213 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2828425 0.79 CNR1 (0.50) CNR1HSP90AA1SRD5A1SRD5A2
SCHEMBL13090171 0.79 CNR1 (0.50) CNR1NPSR1CYP1A2CYP3A4CYP2C9
SCHEMBL4464885 0.75 CNR1 (0.64) CNR1ALDH1A1SRD5A1SRD5A2
SCHEMBL6226020 0.75 CNR1 (0.64) CNR1ALDH1A1SRD5A1SRD5A2
Lithium Ion SCHEMBL4481864 0.74 CNR1 (0.60) CNR1ALDH1A1NPSR1SRD5A1SRD5A2
SCHEMBL763027 0.74 CNR1 (0.46) CNR1NPSR1SRD5A1SRD5A2
SCHEMBL6485133 0.74 AHR (0.48) CNR1HTTSRD5A1SRD5A2
SCHEMBL24824309 0.73 SIRT1 (0.38) CNR1ALDH1A1SIRT1
SCHEMBL4481860 0.73 CNR1 (0.62) CNR1ALDH1A1SRD5A1SRD5A2
SCHEMBL10575187 0.72 TSHR (0.56) CYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7576088-B2 Benzodioxole derivatives HOFFMAN-LA ROCHE INC. (US) 2009-08-18 US disclosed
EP-1532132-B1 NOVEL BENZODIOXOLES HOFFMANN LA ROCHE (CH) 2008-03-19 EP disclosed
US-20050143373-A1 Benzodioxole derivatives ALANINE ALEXANDER (FR) 2005-06-30 US disclosed
US-6900227-B2 Benzodioxole derivatives HOFFMANN-LA ROCHE INC. (US) 2005-05-31 US disclosed
EP-1532132-A1 NOVEL BENZODIOXOLES F.HOFFMANN-LA ROCHE AG (CH) 2005-05-25 EP disclosed
US-20040142922-A1 Benzodioxole derivatives HOFFMANN-LA ROCHE INC. 2004-07-22 US disclosed
WO-2004013120-A1 NOVEL BENZODIOXOLES F. HOFFMANN-LA ROCHE AG (CH) 2004-02-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050143373-A1 Benzodioxole derivatives CNR2, CNR1, GPR119 CNR1 2/4885ALDH1A1 607/4885NPSR1 114/4885
US-20040142922-A1 Benzodioxole derivatives CNR1, CNR2, GPR119 CNR1 1/4885ALDH1A1 299/4885NPSR1 131/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.