SCHEMBL4458392

SCHEMBL4458392

CC(C)c1cc(Cc2cnc(N)nc2N)on1

nearest known ligand 0.53

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
DHFR P00374 2/20 0.51
P2RX3 P56373 2/20 0.49
P2RX2 Q9UBL9 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1794999 0.81 DHFR (0.49) DHFR
SCHEMBL1790427 0.80 ALDH1A1 (0.36) DHFR
SCHEMBL1792738 0.75 IGF1R (0.53)
SCHEMBL1791868 0.73 NOTUM (0.52)
SCHEMBL22277760 0.72 DHFR (0.51) DHFRP2RX3P2RX2
SCHEMBL4472365 0.72 DHFR (0.39) DHFR
SCHEMBL22277341 0.71 DHFR (0.50) DHFRP2RX3P2RX2
SCHEMBL22277732 0.71 DHFR (0.50) DHFRP2RX3P2RX2
SCHEMBL4462541 0.71 DHFR (0.43) DHFR
SCHEMBL4462978 0.71 ALDH1A1 (0.51)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009017838-A2 COMBINATIONS OF JAK-2 INHIBITORS AND OTHER AGENTS EXELIXIS, INC. (US) 2009-02-05 WO claimed