SCHEMBL4458984

SCHEMBL4458984

NCc1c(F)c(F)c(F)c(F)c1F.NCc1ccc(F)cc1F

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.48
AGXT P21549 2/20 0.48
MPO P05164 3/20 0.40
KDM4E B2RXH2 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
ALDH1A1 P00352 1/20 0.39
LOXL2 Q9Y4K0 2/20 0.37
DPP4 P27487 1/20 0.36
DAO P14920 1/20 0.35
HTR2A P28223 4/20 0.34
HTR2C P28335 2/20 0.34
HTR2B P41595 1/20 0.34
TRPM8 Q7Z2W7 1/20 0.34
TAAR1 Q96RJ0 1/20 0.33
MAPK14 Q16539 1/20 0.33
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL113852 0.88 IDO1 (0.59) IDO1AGXTMPOKDM4ESMN1; SMN2
SCHEMBL26625794 0.88 IDO1 (0.59) IDO1AGXTMPOKDM4ESMN1; SMN2
Trifluoroacetic Acid SCHEMBL4243585 0.73 IDO1 (0.44) IDO1AGXTALDH1A1HTR2AHTR2C
SCHEMBL1116576 0.73 IDO1 (0.57) IDO1AGXTMPOKDM4ESMN1; SMN2
SCHEMBL29431834 0.73 IDO1 (0.57) IDO1AGXTMPOKDM4ESMN1; SMN2
SCHEMBL12496555 0.72 MAOB (0.48) IDO1AGXTMPOLOXL2HTR2C
SCHEMBL1398042 0.72 MPO (0.48) IDO1AGXTMPOKDM4ESMN1; SMN2
SCHEMBL28750348 0.72 ADRA2B (0.45) IDO1AGXTKDM4ESMN1; SMN2ALDH1A1
Hydrochloric Acid SCHEMBL2209462 0.71 IDO1 (0.59) IDO1AGXTMPOKDM4ESMN1; SMN2
SCHEMBL554229 0.71 SLC6A2 (0.33) LOXL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0819000-B1 NODULISPORIC ACID DERIVATIVES MERCK & CO INC (US) 2009-07-08 EP disclosed