SCHEMBL4459737

SCHEMBL4459737

NC1=NC(N)(c2ccccc2OC(F)(F)F)NC=C1

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 2/20 0.38
HCAR1 Q9BXC0 1/20 0.32
MPL P40238 1/20 0.32
C1R P00736 1/20 0.31
EPHX2 P34913 1/20 0.31
POLB P06746 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
TRPA1 O75762 1/20 0.30
ALOX5AP P20292 1/20 0.30
FEN1 P39748 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12813182 0.82 BACE1 (0.38) BACE1HCAR1MPL
SCHEMBL1172224 0.76 BACE1 (0.32) BACE1
SCHEMBL1171905 0.74 CTSD (0.40) BACE1
SCHEMBL4458379 0.73 CYP3A4 (0.35) NPSR1
SCHEMBL1172152 0.73 TAAR1 (0.39)
SCHEMBL29974839 0.73 HTT (0.31)
SCHEMBL1171691 0.69 BACE1 (0.41) BACE1
SCHEMBL30157203 0.68 JAK2 (0.31) ALOX5APFEN1
SCHEMBL26922378 0.67 BACE1 (0.33) BACE1MPL
SCHEMBL1171769 0.67 ALDH1A1 (0.41) POLBNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009017838-A2 COMBINATIONS OF JAK-2 INHIBITORS AND OTHER AGENTS EXELIXIS, INC. (US) 2009-02-05 WO disclosed