SCHEMBL4461977

SCHEMBL4461977

NC(=O)c1ccc(F)c([O])c1F

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 1/20 0.47
CES2 O00748 7/20 0.45
CES1 P23141 7/20 0.45
MAP2K2 P36507 1/20 0.41
MAP2K1 Q02750 1/20 0.41
HTR1A P08908 1/20 0.37
ALDH1A1 P00352 2/20 0.35
MAPT P10636 2/20 0.35
KDM4E B2RXH2 1/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CASP1 P29466 1/20 0.35
BCHE P06276 1/20 0.34
KMT2A Q03164 2/20 0.34
ATM Q13315 1/20 0.34
PARP10 Q53GL7 2/20 0.34
PARP15 Q460N3 1/20 0.34
MEN1 O00255 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1003016 0.82 CES2 (0.67) DGAT1CES2CES1MAP2K2MAP2K1
SCHEMBL811064 0.81 DGAT1 (0.52) DGAT1CES2CES1MAP2K2MAP2K1
SCHEMBL201107 0.78 DGAT1 (0.47) DGAT1CES2CES1MAP2K2MAP2K1
SCHEMBL3026191 0.78 DGAT1 (0.47) DGAT1CES2CES1MAP2K2MAP2K1
SCHEMBL5802725 0.77 DGAT1 (0.46) DGAT1CES2CES1MAP2K2MAP2K1
SCHEMBL30827695 0.77 DGAT1 (0.55) DGAT1CES2CES1MAP2K2MAP2K1
SCHEMBL30258821 0.74 CES2 (0.50) DGAT1CES2CES1MAP2K2MAP2K1
SCHEMBL2646259 0.74 CES2 (0.48) DGAT1CES2CES1ALDH1A1MAPT
SCHEMBL4355806 0.74 CES2 (0.50) DGAT1CES2CES1MAP2K2MAP2K1
SCHEMBL1204044 0.74 CES2 (0.50) DGAT1CES2CES1MAP2K2MAP2K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7585869-B2 Substituted heterocylces for the treatment of abnormal cell growth PFIZER, INC. (US) 2009-09-08 US claimed