Chromanone

Chromanone

SCHEMBL4463263

NC(N)=O.O=C1CCOc2ccccc21

nearest known ligand 0.53

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 5/20 0.53
MAOA P21397 1/20 0.53
NOTUM Q6P988 1/20 0.52
GRM5 P41594 4/20 0.50
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
NFKB1 P19838 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
PKM P14618 1/20 0.44
TSHR P16473 1/20 0.44
PIK3CA P42336 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
ITGB2 P05107 1/20 0.40
ICAM1 P05362 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Chromanone SCHEMBL4459476 0.95 GRM5 (0.52) MAOBMAOANOTUMGRM5NPC1
Chromanone SCHEMBL4474722 0.91 GRM5 (0.55) MAOBMAOANOTUMGRM5NPC1
Chromanone SCHEMBL28794 0.91 MAOB (0.56) MAOBMAOANOTUMGRM5NPC1
Chromanone SCHEMBL29384996 0.91 MAOB (0.56) MAOBMAOANOTUMGRM5NPC1
Chromanone SCHEMBL28205525 0.91 MAOB (0.56) MAOBMAOANOTUMGRM5NPC1
Chromanone SCHEMBL29349977 0.89 MAOB (0.55) MAOBMAOANOTUMGRM5NPC1
Chromanone SCHEMBL28463260 0.89 MAOB (0.55) MAOBMAOANOTUMGRM5NPC1
Chromanone SCHEMBL27846233 0.89 MAOB (0.55) MAOBMAOANOTUMGRM5NPC1
Chromanone SCHEMBL30017864 0.89 MAOB (0.55) MAOBMAOANOTUMGRM5NPC1
Chromanone SCHEMBL28719460 0.89 MAOB (0.55) MAOBMAOANOTUMGRM5NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004103985-A2 DERIVATIVES OF FUSAROCHROMANONE AS THERAPEUTIC AGENTS UNIVERSITY OF SOUTH CAROLINA (US) 2004-12-02 WO claimed
US-7598403-B2 Synthesis of chromanones THE UNIVERSITY OF SOUTH CAROLINA RESEARCH FOUNDATION (US) 2009-10-06 US disclosed
US-20070203214-A1 Synthesis Of Chromanones UNIVERSITY OF SOUTH CAROLINA (US) 2007-08-30 US disclosed
WO-2004103985-A2 DERIVATIVES OF FUSAROCHROMANONE AS THERAPEUTIC AGENTS UNIVERSITY OF SOUTH CAROLINA (US) 2004-12-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070203214-A1 Synthesis Of Chromanones MAP3K6, MAP3K8, MAP3K1 MAOB 1582/4885MAOA 1648/4885NOTUM 3467/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.