SCHEMBL4465802

SCHEMBL4465802

Nn1c(S)nnc1-c1ccccc1OC(F)(F)F

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 2/20 0.53
KCNN4 O15554 1/20 0.45
CNR2 P34972 1/20 0.40
PDE2A O00408 1/20 0.39
PDE10A Q9Y233 1/20 0.39
NPC1 O15118 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
SCN9A Q15858 8/20 0.38
KDM4E B2RXH2 1/20 0.38
MAPT P10636 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
POLB P06746 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
TRPA1 O75762 1/20 0.36
S1PR1 P21453 1/20 0.36
ALOX5AP P20292 1/20 0.36
FEN1 P39748 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2889816 0.80 KDM4E (0.52) HSD11B1KCNN4PDE2APDE10ANPC1
SCHEMBL4559681 0.77 MEN1 (0.44) KCNN4NPC1ALDH1A1LMNARAB9A
SCHEMBL4944318 0.74 ALDH1A1 (0.46) HSD11B1KCNN4PDE2APDE10ANPC1
SCHEMBL4349748 0.73 ALDH1A1 (0.47) HSD11B1KCNN4NPC1ALDH1A1LMNA
SCHEMBL4350463 0.73 ALDH1A1 (0.48) KCNN4NPC1ALDH1A1LMNARAB9A
SCHEMBL2747278 0.72 HSD11B1 (0.74) HSD11B1KCNN4CNR2PDE2APDE10A
SCHEMBL4345607 0.71 ALDH1A1 (0.76) HSD11B1PDE2APDE10ANPC1ALDH1A1
SCHEMBL10012799 0.71 HSD11B1 (0.46) HSD11B1KCNN4PDE10ANPC1ALDH1A1
SCHEMBL8627702 0.71 ALDH1A1 (0.46) NPC1ALDH1A1LMNARAB9ASMN1; SMN2
SCHEMBL7701143 0.71 ALDH1A1 (0.50) HSD11B1KCNN4CNR2ALDH1A1SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009094205-A2 3-ARYL-6-ARYL-7H-[1,2,4]TRIAZOLO[3,4-B][1,3,4]THIADIAZINES AND ANALOGS AS ACTIVATORS OF CASPASES AND INDUCERS OF APOPTOSIS AND THE USE THEREOF CYTOVIA, INC. (US) 2009-07-30 WO disclosed