SCHEMBL4470656

SCHEMBL4470656

Brc1cc(Br)c2cccnc2c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.52
CYP1A2 P05177 1/20 0.52
CYP2C19 P33261 1/20 0.52
KDM4E B2RXH2 3/20 0.48
MAPT P10636 3/20 0.48
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
HSP90AA1 P07900 2/20 0.47
USP2 O75604 1/20 0.47
TP53 P04637 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
APAF1 O14727 2/20 0.44
SYK P43405 5/20 0.43
NR4A2 P43354 1/20 0.43
LMNA P02545 2/20 0.42
NQO2 P16083 1/20 0.41
AXL P30530 1/20 0.41
ALK Q9UM73 1/20 0.40
CYP3A4 P08684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29551392 1.00 HTT (0.52) HTTCYP1A2CYP2C19KDM4EMAPT
SCHEMBL116193 0.84 HTT (0.48) HTTCYP1A2CYP2C19KDM4EMAPT
SCHEMBL23619926 0.80 NR4A2 (0.49) HTTCYP1A2CYP2C19KDM4EMAPT
SCHEMBL30908153 0.80 ALDH1A1 (0.48) HTTCYP1A2CYP2C19KDM4EMAPT
SCHEMBL31606740 0.80 NR4A2 (0.62) HTTCYP1A2CYP2C19KDM4EMAPT
SCHEMBL3454205 0.80 NR4A2 (0.49) HTTCYP1A2CYP2C19KDM4EMAPT
SCHEMBL3711428 0.80 KDM4E (0.45) HTTCYP1A2CYP2C19KDM4EMAPT
SCHEMBL18318260 0.80 ALDH1A1 (0.48) HTTCYP1A2CYP2C19KDM4EMAPT
SCHEMBL22719670 0.80 KDM4E (0.53) HTTCYP1A2CYP2C19KDM4EMAPT
SCHEMBL14659006 0.80 HTT (0.48) HTTCYP1A2CYP2C19KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 37 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112457243-B Synthesis method of 7-bromo-5-methoxyquinoline 苏州康润医药有限公司 2022-04-12 CN claimed
CN-112457243-A Synthesis method of 7-bromo-5-methoxyquinoline 苏州康润医药有限公司 2021-03-09 CN claimed
CN-110041905-B Fluorescent and phosphorescent dual luminescent material with switching effect and preparation method thereof 华中科技大学 2020-05-19 CN claimed
WO-2009140215-A2 METHOD FOR TREATING DRUG-RESISTANT BACTERIAL AND OTHER INFECTIONS WITH CLIOQUINOL, PHANQUINONE, AND RELATED COMPOUNDS GERAGHTY, ERIN (US) 2009-11-19 WO claimed
US-20080207673-A1 Method for Treating Cancer, Coronary, Inflammatory and Macular Disease, Combining the Modulation of Zinc-and/or Copper Dependent Proteins XILINAS MICHEL 2008-08-28 US claimed
WO-2006117660-A2 METHOD FOR TREATING CANCER, CORONARY, INFLAMMATORY AND MACULAR DISEASE, COMBINING THE MODULATION OF ZINC- AND/OR COPPER DEPENDENT PROTEINS CLIO PHARMACEUTICAL CORPORATION (US) 2006-11-09 WO claimed
EP-4079724-B1 2-(2-CHLOROPHENYL)-N-(5-SULFAMOYLISOQUINOLIN-7-YL)ACETAMIDE DERIVATIVES AND SIMILAR COMPOUNDS AS P2X4 ANTAGONISTS FOR THE TREATMENT OF E.G. URINARY TRACT DISEASES WUHAN LL SCIENCE & TECHNOLOGY DEVELOPMENT CO LTD (CN) 2025-11-12 EP disclosed
US-20250025443-A1 COMPOUNDS AND METHODS FOR TREATING CORONA VIRUSES Clear Creek Bio, Inc. (US) 2025-01-23 US disclosed
CN-114901642-B Fused ring compound and application thereof 武汉朗来科技发展有限公司 2024-02-23 CN disclosed
WO-2023064493-A1 COMPOUNDS AND METHODS FOR TREATING CORONAVIRUSES Clear Creek Bio, Inc. (US) 2023-04-20 WO disclosed
WO-2023064493-A1 COMPOUNDS AND METHODS FOR TREATING CORONAVIRUSES Clear Creek Bio, Inc. (US) 2023-04-20 WO disclosed
US-20230118751-A1 FUSED RING COMPOUND AND APPLICATION THEREOF WUHAN LL SCIENCE AND TECHNOLOGY DEVELOPMENT CO., LTD. (CN) 2023-04-20 US disclosed
US-20230118751-A1 FUSED RING COMPOUND AND APPLICATION THEREOF WUHAN LL SCIENCE AND TECHNOLOGY DEVELOPMENT CO., LTD. (CN) 2023-04-20 US disclosed
WO-2006117660-A2 METHOD FOR TREATING CANCER, CORONARY, INFLAMMATORY AND MACULAR DISEASE, COMBINING THE MODULATION OF ZINC- AND/OR COPPER DEPENDENT PROTEINS CLIO PHARMACEUTICAL CORPORATION (US) 2006-11-09 WO disclosed
WO-2002051415-A2 USE OF SEQUESTRANTS FOR TREATING PRION DISEASES XILINAS MICHEL (CY) 2002-07-04 WO disclosed
EP-0138773-B1 USE OF QUINOLINE DERIVATIVES FOR THE PROTECTION OF CROP PLANTS CIBA-GEIGY AG (CH) 1990-08-29 EP disclosed
US-4749406-A Quinoline derivatives and compositions thereof for the protection of cultivated plants CIBA-GEIGY CORPORATION (US) 1988-06-07 US disclosed
US-4585472-A PRE- AND POSTEMERGENCE HERBICIDES BASF AKTIENGESELLSCHAFT (DE) 1986-04-29 US disclosed
EP-0138773-A2 Use of quinoline derivatives for the protection of crop plants CIBA-GEIGY AG (CH) 1985-04-24 EP disclosed
EP-0102542-A2 1,2,4,6-Thiatriazin-1,1-dioxide ethers, process for their preparation and their use as herbicides BASF Aktiengesellschaft (DE) 1984-03-14 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230118751-A1 FUSED RING COMPOUND AND APPLICATION THEREOF P2RX4, P2RX3, P2RX2 HTT 2671/4885CYP1A2 657/4885CYP2C19 517/4885
US-20250025443-A1 COMPOUNDS AND METHODS FOR TREATING CORONA VIRUSES ACE, PREP, PEPD HTT 2553/4885CYP1A2 2421/4885CYP2C19 1297/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.