SCHEMBL4470741

SCHEMBL4470741

COc1cncnc1N1CCN(CCCc2c[nH]c3ccc(N)cc23)CC1.O=[N+]([O-])c1ccc2[nH]cc(CCCBr)c2c1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 12/20 0.43
SLC6A4 P31645 1/20 0.43
HTR7 P34969 1/20 0.43
KCNH2 Q12809 1/20 0.43
ADRA2A P08913 1/20 0.41
ADRA2B P18089 1/20 0.41
ADRA2C P18825 1/20 0.41
ADRA1D P25100 1/20 0.41
ADRA1A P35348 1/20 0.41
ADRA1B P35368 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4347857 0.92 HTR1A (0.50) HTR1ASLC6A4HTR7KCNH2ADRA2A
SCHEMBL4353460 0.88 HTR1A (0.54) HTR1ASLC6A4HTR7KCNH2ADRA2A
SCHEMBL9373347 0.80 HTR1A (0.69) HTR1AADRA2AADRA2BADRA2CADRA1D
SCHEMBL8824019 0.79 HTR1A (0.57) HTR1ASLC6A4HTR7KCNH2ADRA2A
SCHEMBL4357142 0.79 HTR1A (0.68) HTR1ASLC6A4HTR7KCNH2
SCHEMBL6354737 0.79 HTR1A (0.66) HTR1ASLC6A4HTR7KCNH2ADRA2A
SCHEMBL4347602 0.79 HTR1A (0.54) HTR1ASLC6A4HTR7KCNH2ADRA2A
SCHEMBL4349471 0.79 ADRA2A (0.63) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL8978667 0.78 HTR1A (0.48) HTR1ASLC6A4HTR7KCNH2ADRA2A
Hydrochloric Acid SCHEMBL4356376 0.78 HTR1A (0.70) HTR1ASLC6A4HTR7KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009137733-A1 INDOLYLALKYL DERIVATIVES OF PYRIMIDINYLPIPERAZINE AND METABOLITES THEREOF FOR TREATMENT OF ANXIETY, DEPRESSION, AND SEXUAL DYSFUNCTION FABRE-KRAMER PHARMACEUTICALS, INC. (US) 2009-11-12 WO disclosed