SCHEMBL4471205

SCHEMBL4471205

COc1ccc(CNCCNC(=O)c2cccc(C(=O)NCCN3CCC(OC(=O)N(c4ccccc4-c4ccccc4)N(C(=O)O)c4ccccc4-c4ccccc4)CC3)c2)cc1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CCR3 P51677 2/20 0.46
DRD4 P21917 8/20 0.43
ADRB2 P07550 2/20 0.42
CHRM3 P20309 2/20 0.42
SLC5A7 Q9GZV3 1/20 0.42
DRD2 P14416 2/20 0.42
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
SLC6A2 P23975 1/20 0.41
SLC6A4 P31645 1/20 0.41
PLD2 O14939 1/20 0.40
PLD1 Q13393 1/20 0.40
CACNA1G O43497 1/20 0.40
CARM1 Q86X55 1/20 0.40
PRMT6 Q96LA8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4494191 0.93 CHRM2 (0.43) CCR3DRD4ADRB2CHRM3SLC5A7
SCHEMBL4471210 0.92 CCR3 (0.48) CCR3DRD4ADRB2CHRM3SLC5A7
SCHEMBL4494194 0.87 CCR3 (0.43) CCR3DRD4ADRB2CHRM3SLC5A7
SCHEMBL4475332 0.86 ADRB2 (0.43) ADRB2CHRM3SLC5A7CARM1PRMT6
SCHEMBL4487266 0.86 ADRB2 (0.49) CCR3DRD4ADRB2CHRM3DRD2
SCHEMBL4483079 0.86 CHRM3 (0.44) ADRB2CHRM3SLC5A7DRD2CARM1
SCHEMBL265292 0.85 CHRM3 (0.56) ADRB2CHRM3
SCHEMBL4484438 0.84 CHRM3 (0.43) ADRB2CHRM3DRD2
SCHEMBL4494455 0.84 CHRM2 (0.43) ADRB2CHRM3DRD2
SCHEMBL4493963 0.83 CHRM3 (0.45) ADRB2CHRM3SLC5A7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7632847-B2 Bronchodilators; treating chronic obstructive pulmonary disease or asthma; long duration of action; reduced side effects, such as dry-mouth and constipation; e.g. biphenyl-2-ylcarbamic acid 1-(2-(3-[3-(4-hydroxybenzylamino)propionylamino]benzoylamino)ethyl)piperidin-4-yl ester THERAVANCE, INC. (US) 2009-12-15 US disclosed