SCHEMBL4472407

SCHEMBL4472407

COC(=O)C(N)Cc1ccc(OC(C)(C)C)cc1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACACB O00763 4/20 0.53
PTPN1 P18031 1/20 0.50
ALDH1A1 P00352 1/20 0.46
PTGS2 P35354 1/20 0.45
LTA4H P09960 1/20 0.44
LDHA P00338 1/20 0.41
KIF11 P52732 1/20 0.41
ESR1 P03372 1/20 0.41
ESR2 Q92731 1/20 0.41
SLC6A4 P31645 1/20 0.40
CTSL P07711 1/20 0.40
CTSK P43235 1/20 0.40
ITGB3 P05106 1/20 0.40
ITGA2B P08514 1/20 0.40
PPARG P37231 1/20 0.40
PPARA Q07869 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2058886 1.00 ACACB (0.53) ACACBPTPN1ALDH1A1PTGS2LTA4H
Hydrochloric Acid SCHEMBL1310837 0.98 ACACB (0.52) ACACBPTPN1ALDH1A1PTGS2LTA4H
Hydrochloric Acid SCHEMBL1310835 0.98 ACACB (0.52) ACACBPTPN1ALDH1A1PTGS2LTA4H
SCHEMBL2311154 0.88 ACACB (0.50) ACACBPTPN1LTA4HLDHACTSL
SCHEMBL2311151 0.88 ACACB (0.50) ACACBPTPN1LTA4HLDHACTSL
SCHEMBL3729750 0.88 ACACB (0.50) ACACBPTPN1LTA4HLDHACTSL
SCHEMBL16080173 0.88 ACACB (0.50) ACACBPTPN1LTA4HLDHACTSL
Hydrochloric Acid SCHEMBL3745279 0.87 ACACB (0.49) ACACBPTPN1ALDH1A1LTA4HLDHA
SCHEMBL8751946 0.87 ACACB (0.49) ACACBPTPN1LTA4HLDHACTSL
Hydrochloric Acid SCHEMBL29398263 0.87 ACACB (0.49) ACACBPTPN1ALDH1A1LTA4HLDHA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110082087-A1 COMPOUNDS FOR TREATING PAIN Edificio ICAT (PT) 2011-04-07 US disclosed
US-20110082087-A1 COMPOUNDS FOR TREATING PAIN Edificio ICAT (PT) 2011-04-07 US disclosed
WO-2009123487-A1 COMPOUNDS FOR TREATING PAIN BIOALVO - SERVIÇOS, INVESTIGAÇÃO E DESENVOLVIMENTO EM BIOTECNOLOGIA S.A. (PT) 2009-10-08 WO disclosed
US-7511063-B2 High affinity quinoline-based kinase ligands SCHERING CORPORATION (US) 2009-03-31 US disclosed
US-20080045568-A1 Novel high affinity quinoline-based kinase ligands SCHERING CORPORATION 2008-02-21 US disclosed
US-6423689-B1 Peptidyl calcium channel blockers WARNER-LAMBERT COMPANY 2002-07-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080045568-A1 Novel high affinity quinoline-based kinase ligands CDKL2, CDK2, CDKL1 ACACB 2110/4885PTPN1 2030/4885ALDH1A1 4640/4885
US-20110082087-A1 COMPOUNDS FOR TREATING PAIN PTGS2, CNR2, PTGS1 ACACB 1199/4885PTPN1 3524/4885ALDH1A1 1297/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.