Nogalamycin

Nogalamycin

SCHEMBL4473

COC(=O)[C@@H]1c2cc3c(c(O)c2[C@@H](O[C@@H]2O[C@@H](C)[C@H](OC)[C@@](C)(OC)[C@H]2OC)C[C@]1(C)O)C(=O)c1c(O)cc2c(c1C3=O)OC1O[C@@]2(C)[C@H](O)[C@@H](N(C)C)[C@@H]1O

nearest known ligand 0.72

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 3/20 0.72
ALDH1A1 P00352 2/20 0.72
CYP1A2 P05177 2/20 0.72
HPGD P15428 2/20 0.72
ALOX15 P16050 2/20 0.72
CYP2D6 P10635 1/20 0.72
MEN1 O00255 3/20 0.45
USP2 O75604 3/20 0.45
MAPT P10636 3/20 0.45
KMT2A Q03164 3/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
KDM4E B2RXH2 2/20 0.45
THRB P10828 2/20 0.45
BLM P54132 2/20 0.45
CASP1 P29466 1/20 0.45
TP53 P04637 2/20 0.41
CYP3A4 P08684 2/20 0.41
RECQL P46063 2/20 0.41
HBB P68871 2/20 0.41
RGS12 O14924 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Nogalamycin SCHEMBL4472 1.00 HSD17B10 (0.72) HSD17B10ALDH1A1CYP1A2HPGDALOX15
Nogalamycin SCHEMBL29356331 1.00 HSD17B10 (0.72) HSD17B10ALDH1A1CYP1A2HPGDALOX15
Nogalamycin SCHEMBL1649692 1.00 HSD17B10 (0.72) HSD17B10ALDH1A1CYP1A2HPGDALOX15
Nogalamycinic Acid SCHEMBL30055177 0.95 HSD17B10 (0.65) HSD17B10ALDH1A1CYP1A2HPGDALOX15
SCHEMBL18567081 0.91 HSD17B10 (0.72) HSD17B10ALDH1A1CYP1A2HPGDALOX15
Disnogamycin SCHEMBL29390994 0.88 HSD17B10 (0.55) HSD17B10ALDH1A1CYP1A2HPGDALOX15
Disnogamycin SCHEMBL26459009 0.88 HSD17B10 (0.55) HSD17B10ALDH1A1CYP1A2HPGDALOX15
SCHEMBL3345418 0.84 HSD17B10 (1.00) HSD17B10ALDH1A1CYP1A2HPGDALOX15
SCHEMBL11468050 0.84 HSD17B10 (1.00) HSD17B10ALDH1A1CYP1A2HPGDALOX15
SCHEMBL18593716 0.77 HSD17B10 (0.52) HSD17B10ALDH1A1CYP1A2HPGDALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 32173 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4748859-A2 CHEMICALLY AND PHOTOCHEMICALLY INITIATED CELL MEMBRANE BLEBBING TO INDUCE CELL VESICLE PRODUCTION, MODIFICATIONS THEREOF, AND USES THEREOF The Regents of the University of California (US) 2026-05-27 EP claimed
EP-4743490-A1 HUMANIZED ANTI-CD7 ANTIBODY Christian-Albrechts-Universität zu Kiel (DE) 2026-05-20 EP claimed
WO-2026099502-A1 NOVEL DRUG CONJUGATES FOR TESTING CELLULAR DRUG UPTAKE Deutsches Krebsforschungszentrum Stiftung des öffentlichen Rechts (DE) 2026-05-15 WO claimed
US-20260115305-A1 LINKERS, CONJUGATES AND APPLICATIONS THEREOF GENEQUANTUM HEALTHCARE SUZHOU CO LTD (CN) 2026-04-30 US claimed
US-20260116861-A1 ISOXAZOLE HYDROXAMIC ACIDS AS HISTONE DEACETYLASE 6 INHIBITORS THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-04-30 US claimed
US-20260108619-A1 CONJUGATION LINKERS, CELL BINDING MOLECULE-DRUG CONJUGATES CONTAINING THE LINKERS, METHODS OF MAKING AND USES SUCH CONJUGATES WITH THE LINKERS HANGZHOU DAC BIOTECH CO., LTD. (CN) 2026-04-23 US claimed
US-20260085100-A1 METHODS OF ANTIGEN PRODUCTION THE WISTAR INSTITUTE OF ANATOMY AND BIOLOGY (US) 2026-03-26 US claimed
US-20260077056-A1 LINKER-PAYLOAD COMPOUND, CONJUGATES AND APPLICATIONS THEREOF GENEQUANTUM HEALTHCARE SUZHOU CO LTD (CN) 2026-03-19 US claimed
US-12576124-B2 Formulation of a conjugate of a tubulysin analog to a cell-binding molecule HANGZHOU DAC BIOTECH CO., LTD (CN) 2026-03-17 US claimed
EP-4698185-A1 METHODS AND SYSTEMS FOR IMPROVING ANTI-CANCER THERAPIES Osasuna Therapeutics SA (CH) 2026-02-25 EP claimed
WO-2000028087-A1 A LIBRARY OF MODIFIED PRIMERS FOR NUCLEIC ACID SEQUENCING, AND METHOD OF USE THEREOF SEQUETECH CORPORATION (US) 2000-05-18 WO claimed
EP-1000078-A1 HYBRID ANTHRACYCLINES FROM GENETICALLY ENGINEERED $i(STREPTOMYCES GALILAEUS) STRAINS GALILAEUS OY (FI) 2000-05-17 EP claimed
WO-1999058126-B1 USE OF NEOMYCIN FOR TREATING ANGIOGENESIS-RELATED DISEASES ENDOWMENT RES INHUMAN BIOLOGY (US) 2000-02-17 WO claimed
WO-1999058544-A9 HYBRID ANTHRACYCLINES FROM GENETICALLY ENGINEERED STREPTOMYCES GALILAEUS STRAINS GALILAEUS OY (FI) 2000-01-20 WO claimed
WO-1999058544-A1 HYBRID ANTHRACYCLINES FROM GENETICALLY ENGINEERED STREPTOMYCES GALILAEUS STRAINS GALILAEUS OY (FI) 1999-11-18 WO claimed
WO-1999058126-A1 USE OF NEOMYCIN FOR TREATING ANGIOGENESIS-RELATED DISEASES THE ENDOWMENT FOR RESEARCH IN HUMAN BIOLOGY, INC. (US) 1999-11-18 WO claimed
EP-0316440-B1 System and method for providing localized Mössbauer absorption in an organic medium MILLS RANDELL L (US) 1996-01-03 EP claimed
WO-1994026253-A1 LIPOSOME HAVING A MULTICOMPONENT BILAYER WHICH CONTAINS A BIOACTIVE AGENT AS AN INTEGRAL COMPONENT OF THE BILAYER THE LIPOSOME COMPANY, INC. (US) 1994-11-24 WO claimed
WO-1992005200-A1 XENOBIOTIC-ANTIBODY CONJUGATES CHEMEX PHARMACEUTICALS, INC. (US) 1992-04-02 WO claimed
US-4329450-A Nogalamycin analog containing compounds THE UPJOHN COMPANY (US) 1982-05-11 US claimed