SCHEMBL4474261

SCHEMBL4474261

COc1[c]cc(OC(F)(F)F)c(OC)c1

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 1/20 0.33
KCNK9 Q9NPC2 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
CYP3A4 P08684 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL592705 0.82 CYP3A4 (0.39) CYP1A2CYP2C9CYP2C19CYP3A4MAPT
SCHEMBL7945837 0.80
SCHEMBL10829023 0.76 HTR2A (0.41) MAPT
SCHEMBL3279036 0.76 HTR2A (0.41) CYP3A4MAPT
SCHEMBL28188574 0.72 LMNA (0.36) CYP3A4MAPT
SCHEMBL7255898 0.72 ACHE (0.33) CYP3A4MAPT
SCHEMBL1637863 0.70 ACHE (0.39) CYP3A4MAPT
SCHEMBL1969378 0.70 ACHE (0.39) CYP3A4MAPT
SCHEMBL5090699 0.68 POLB (0.39) MAPT
SCHEMBL21830291 0.68 PDE4A (0.42) CYP1A2CYP2C9CYP2C19CYP3A4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7598274-B2 N-methyl-4-{4-[5-(4-chloro-3-trifluoromethylphenylcarbamoyl)-1H-pyrrol-3-yl]-phenoxy}pyridine-2-carboxamide; Raf kinases inhibitors MERCK PATENT GMBH (DE) 2009-10-06 US claimed