SCHEMBL4479047

SCHEMBL4479047

c1cnc([C@H]2c3ccc(OC4CCN(C5CCC5)CC4)cc3CC23CCNCC3)cn1

nearest known ligand 0.46

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 20/20 0.46
KCNH2 Q12809 4/20 0.41
CYP2D6 P10635 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4478245 0.76 HRH3 (0.48) HRH3KCNH2CYP2D6
SCHEMBL4474695 0.74 HRH3 (0.48) HRH3
SCHEMBL3776595 0.73 HRH3 (0.62) HRH3KCNH2CYP2D6
SCHEMBL4485943 0.72 HRH3 (0.45) HRH3KCNH2CYP2D6
SCHEMBL3766350 0.71 HRH3 (0.46) HRH3KCNH2CYP2D6
SCHEMBL3094888 0.67 HRH3 (0.64) HRH3CYP2D6
SCHEMBL3085867 0.65 HRH3 (1.00) HRH3CYP2D6
SCHEMBL3091232 0.64 HRH3 (0.68) HRH3CYP2D6
SCHEMBL11918570 0.62 HRH3 (1.00) HRH3KCNH2CYP2D6
SCHEMBL3077588 0.62 HRH3 (0.95) HRH3CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009039431-A2 SUBSTITUTED ARYL-FUSED SPIROCYCLIC AMINES NEUROGEN CORPORATION (US) 2009-03-26 WO claimed