SCHEMBL4480672

SCHEMBL4480672

CCOC(=O)C1CCCC1N(CCN(C)C)C(=O)CC1=NS(=O)(=O)c2cc(NS(C)(=O)=O)ccc2N1

nearest known ligand 0.32

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 1/20 0.31
MMP13 P45452 1/20 0.31
RECQL P46063 2/20 0.31
LMNA P02545 3/20 0.31
ALDH1A1 P00352 2/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
THRB P10828 1/20 0.30
HPGD P15428 1/20 0.30
TP53 P04637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4493109 0.93 MMP2 (0.33) MMP2MMP13RECQLLMNAALDH1A1
SCHEMBL4489808 0.92 MMP2 (0.31) MMP2MMP13RECQLLMNAALDH1A1
SCHEMBL13712260 0.92 MMP2 (0.31) MMP2MMP13RECQLLMNAALDH1A1
SCHEMBL4491594 0.91 MMP2 (0.31) MMP2MMP13RECQLLMNAALDH1A1
SCHEMBL4495276 0.91 MMP2 (0.31) MMP2MMP13RECQLLMNAALDH1A1
SCHEMBL13712254 0.91 MMP2 (0.31) MMP2MMP13RECQLLMNAALDH1A1
SCHEMBL13712257 0.91 MMP2 (0.31) MMP2MMP13RECQLLMNAALDH1A1
SCHEMBL4490615 0.90 MMP2 (0.33) MMP2MMP13RECQLLMNAALDH1A1
SCHEMBL4493945 0.90 MMP2 (0.31) MMP2MMP13RECQLLMNAALDH1A1
SCHEMBL13712266 0.90 MMP2 (0.31) MMP2MMP13RECQLLMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582626-B2 5,6-dihydro-1H-pyridin-2-one compounds ANADYS PHARMACEUTICALS, INC. (US) 2009-09-01 US disclosed
US-7582626-B2 5,6-dihydro-1H-pyridin-2-one compounds ANADYS PHARMACEUTICALS, INC. (US) 2009-09-01 US disclosed
US-7582626-B2 5,6-dihydro-1H-pyridin-2-one compounds ANADYS PHARMACEUTICALS, INC. (US) 2009-09-01 US disclosed
US-20090111798-A1 5,6-DIHYDRO-1H-PYRIDIN-2-ONE COMPOUNDS ANADYS PHARMACEUTICALS, INC. 2009-04-30 US disclosed
US-20090111798-A1 5,6-DIHYDRO-1H-PYRIDIN-2-ONE COMPOUNDS ANADYS PHARMACEUTICALS, INC. 2009-04-30 US disclosed
US-20090111798-A1 5,6-DIHYDRO-1H-PYRIDIN-2-ONE COMPOUNDS ANADYS PHARMACEUTICALS, INC. 2009-04-30 US disclosed
WO-2008073982-A2 5,6-DIHYDRO-1H-PYRIDIN-2-ONE COMPOUNDS ANADYS PHARMACEUTICALS, INC. (US) 2008-06-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090111798-A1 5,6-DIHYDRO-1H-PYRIDIN-2-ONE COMPOUNDS HAVCR2, PYGL, HCCS MMP2 4305/4885MMP13 3395/4885RECQL 446/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.