SCHEMBL4484308

SCHEMBL4484308

Cc1[nH]c(C)c(-c2ccc(-c3cccc(Cl)c3)nc2)c(=O)c1Br

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 2/20 0.48
MAPT P10636 2/20 0.40
KMT2A Q03164 2/20 0.40
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
KDM1A O60341 1/20 0.39
MAOB P27338 1/20 0.39
GRIN2D O15399 1/20 0.37
GRIN3B O60391 1/20 0.37
GRIN1 Q05586 1/20 0.37
GRIN2A Q12879 1/20 0.37
GRIN2B Q13224 1/20 0.37
GRIN2C Q14957 1/20 0.37
GRIN3A Q8TCU5 1/20 0.37
IDO1 P14902 1/20 0.37
IKBKE Q14164 1/20 0.37
PIN1 Q13526 1/20 0.37
CDC7 O00311 1/20 0.36
MEN1 O00255 1/20 0.36
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4490539 0.88 KDM1A (0.41) SLC2A1MAPTKMT2ALMNASMN1; SMN2
SCHEMBL4487868 0.87 SLC2A1 (0.45) SLC2A1MAPTKMT2ASMN1; SMN2KDM1A
SCHEMBL4490477 0.85 SLC2A1 (0.48) SLC2A1MAPTKMT2AMEN1
SCHEMBL4493390 0.83 SLC2A1 (0.66) SLC2A1KDM1AMAOBGRIN1GRIN2B
SCHEMBL4475105 0.83 SLC2A1 (0.53) SLC2A1CHEK1HSD17B1HSD17B2
SCHEMBL4488013 0.80 SLC2A1 (0.45) SLC2A1KMT2ALMNAGRIN2DGRIN3B
SCHEMBL4464652 0.79 SLC2A1 (0.47) SLC2A1
SCHEMBL4475947 0.78 SLC2A1 (0.43) SLC2A1MAPT
SCHEMBL13754689 0.77 BRD4 (0.47) SLC2A1MAPTKMT2ALMNASMN1; SMN2
SCHEMBL4487292 0.77 SLC2A1 (0.44) SLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7579353-B2 Pyridinone derivatives against malaria GLAXO GROUP LIMITED (GB) 2009-08-25 US claimed
US-20080287461-A1 Pyridinone Derivatives Against Malaria GLAXO GROUP LIMITED (GB) 2008-11-20 US claimed
US-7579353-B2 Pyridinone derivatives against malaria GLAXO GROUP LIMITED (GB) 2009-08-25 US disclosed
US-7579353-B2 Pyridinone derivatives against malaria GLAXO GROUP LIMITED (GB) 2009-08-25 US disclosed
US-7579353-B2 Pyridinone derivatives against malaria GLAXO GROUP LIMITED (GB) 2009-08-25 US disclosed
US-20080287461-A1 Pyridinone Derivatives Against Malaria GLAXO GROUP LIMITED (GB) 2008-11-20 US disclosed
US-20080287461-A1 Pyridinone Derivatives Against Malaria GLAXO GROUP LIMITED (GB) 2008-11-20 US disclosed
US-20080287461-A1 Pyridinone Derivatives Against Malaria GLAXO GROUP LIMITED (GB) 2008-11-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080287461-A1 Pyridinone Derivatives Against Malaria G6PD, PNPO, PLPBP SLC2A1 2278/4885MAPT 1942/4885KMT2A 3141/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.