SCHEMBL4484350

SCHEMBL4484350

COc1cc(Cl)c(S(=O)(=O)CNCCOCC(=O)O)c(Cl)c1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.36
KDM4E B2RXH2 3/20 0.36
LMNA P02545 2/20 0.33
TSHR P16473 3/20 0.33
ALDH1A1 P00352 2/20 0.33
GAA P10253 2/20 0.32
MARS1 P56192 1/20 0.32
DDR1 Q08345 1/20 0.32
POLB P06746 1/20 0.32
HTT P42858 2/20 0.32
NPSR1 Q6W5P4 1/20 0.32
MCL1 Q07820 1/20 0.32
PDCD1LG2 Q9BQ51 1/20 0.32
CD274 Q9NZQ7 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
FLT1 P17948 1/20 0.32
FLT4 P35916 1/20 0.32
KDR P35968 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL493564 0.87 TDP1 (0.36) TDP1KDM4ELMNATSHR
SCHEMBL571406 0.86 BDKRB1 (0.37) TDP1KDM4ETSHRGAAPOLB
SCHEMBL15347788 0.85 BDKRB1 (0.37) TDP1KDM4ETSHRGAAPOLB
SCHEMBL5117767 0.85 TDP1 (0.42) TDP1KDM4ELMNATSHRALDH1A1
SCHEMBL4475594 0.85 KDM4E (0.40) TDP1KDM4ETSHRALDH1A1GAA
SCHEMBL493617 0.82 KMT2A (0.42) LMNAALDH1A1GAAPOLBPDCD1LG2
SCHEMBL5130040 0.82 MEN1 (0.39) TDP1KDM4ELMNATSHRHTT
SCHEMBL4000802 0.80 KMT2A (0.40) TDP1TSHRALDH1A1GAADDR1
SCHEMBL493486 0.79 HTT (0.52) TDP1ALDH1A1HTTNPSR1
SCHEMBL4461535 0.77 FABP4 (0.43) KDM4ELMNAALDH1A1POLBHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7538111-B2 Benzenesulphonamide derivatives, method for production and use thereof for treatment of pain LABORATOIRES FOURNIER S.A. (FR) 2009-05-26 US disclosed
US-20060178360-A1 Benzenesulphonamide derivatives, method for production and use thereof for treatment of pain LABORATOIRES FOURNIER S.A. (FR) 2006-08-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060178360-A1 Benzenesulphonamide derivatives, method for production and use thereof for treatment of pain LTB4R2, BDKRB2, TBXA2R TDP1 3724/4885KDM4E 2998/4885LMNA 3898/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.