SCHEMBL4488472

SCHEMBL4488472

CCOC(=O)c1ccc(-c2n[nH]c3ccccc23)cc1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.74
MAP2K4 P45985 4/20 0.63
RAB9A P51151 3/20 0.54
ALDH1A1 P00352 2/20 0.54
MAPT P10636 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
MEN1 O00255 1/20 0.54
HCRTR1 O43613 1/20 0.54
KMT2A Q03164 1/20 0.54
MAPK1 P28482 2/20 0.53
MAPK8 P45983 2/20 0.53
F2RL3 Q96RI0 1/20 0.53
RARA P10276 1/20 0.52
RARB P10826 1/20 0.52
RARG P13631 1/20 0.52
MAPK10 P53779 2/20 0.51
GAA P10253 2/20 0.51
ALPL P05186 1/20 0.51
IDO1 P14902 1/20 0.51
HPGD P15428 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27496466 0.86 MAP2K4 (0.66) KDM4EMAP2K4RAB9AALDH1A1MAPT
SCHEMBL8126956 0.85 MAPK1 (0.72) KDM4EMAP2K4RAB9AALDH1A1SMN1; SMN2
SCHEMBL8681986 0.84 KDM4E (0.60) KDM4EMAP2K4RAB9AALDH1A1MAPT
SCHEMBL11903949 0.81 MAP2K4 (0.63) KDM4EMAP2K4RAB9AALDH1A1MAPK1
SCHEMBL21802593 0.80 KDM4E (0.56) KDM4EMAP2K4RAB9AALDH1A1MAPT
SCHEMBL4119529 0.80 ITK (0.62) KDM4ERAB9AALDH1A1MAPTSMN1; SMN2
SCHEMBL5386371 0.80 ALOX5 (0.55) KDM4EMAP2K4RAB9AALDH1A1MAPT
SCHEMBL27956842 0.79 MAP2K4 (0.60) KDM4EMAP2K4RAB9AALDH1A1MAPK1
SCHEMBL959364 0.79 KDM4E (1.00) KDM4ERAB9AALDH1A1MAPTSMN1; SMN2
SCHEMBL29709972 0.79 KDM4E (1.00) KDM4ERAB9AALDH1A1MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100516049-C Antiangiogenic agent N2Synthesis of- (substituted arylmethyl) -3- (substituted phenyl) indazoles YUNG SHIN PHARM IND CO LTD (CN) 2009-07-22 CN disclosed
US-7514465-B2 Synthesis of N2-(substituted arylmethyl)-3-(substituted phenyl)indazoles as novel anti-angiogenic agents YUNG SHIN PHARM. IND. CO., LTD. (TW) 2009-04-07 US disclosed
CN-1962640-A Novel anti-angiogenic drug N2Synthesis of- (substituted arylmethyl) -3- (substituted phenyl) indazoles YUNG SHIN PHARM IND CO LTD (CN) 2007-05-16 CN disclosed
EP-1659115-A1 Synthesis of substituted 2H-indazole derivatives as anti-angiogenic agents Yung Shin Pharm. Ind. Co., Ltd. (TW) 2006-05-24 EP disclosed
US-20060106032-A1 Synthesis of N2 - (substituted arylmethyl) -3- (substituted phenyl) indazoles as novel anti-angiogenic agents YUNG SHIN PHARM. IND. CO., LTD. (TW) 2006-05-18 US disclosed
CN-1215060-C Fused pyrazolyl compounds, compositions containing the same, and uses of the compounds YONGXIN MEDICINE INDUSTRY CO L (CN) 2005-08-17 CN disclosed
CN-1331076-A Fused pyrazolyl compounds, compositions containing the same, and uses of the compounds YONGXIN MEDICINE INDUSTRY CO L (CN) 2002-01-16 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060106032-A1 Synthesis of N2 - (substituted arylmethyl) -3- (substituted phenyl) indazoles as novel anti-angiogenic agents FLT4, FLT1, KDR KDM4E 1210/4885MAP2K4 1359/4885RAB9A 3692/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.