SCHEMBL4488787

SCHEMBL4488787

O=c1cc(OS(=O)(=O)C(F)(F)F)c2ncccc2n1OCc1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.40
TSHR P16473 2/20 0.40
OPRM1 P35372 1/20 0.39
OPRD1 P41143 1/20 0.39
KDM4E B2RXH2 5/20 0.38
HSD17B10 Q99714 2/20 0.38
ALOX15 P16050 1/20 0.36
PDE4A P27815 3/20 0.35
PDE4C Q08493 3/20 0.35
PDE4D Q08499 3/20 0.35
SLC40A1 Q9NP59 1/20 0.35
NPSR1 Q6W5P4 3/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
MAPT P10636 3/20 0.34
ESR2 Q92731 1/20 0.33
HBB P68871 1/20 0.33
LMNA P02545 2/20 0.33
PDE10A Q9Y233 1/20 0.32
L3MBTL1 Q9Y468 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3515445 0.83 OPRM1 (0.35) ALDH1A1TSHROPRM1OPRD1KDM4E
SCHEMBL23292260 0.78 PDE4A (0.39) ALDH1A1TSHRPDE4APDE4CPDE4D
SCHEMBL29922710 0.78 PDE4A (0.39) ALDH1A1TSHRPDE4APDE4CPDE4D
SCHEMBL16274844 0.74 ESR2 (0.36) ALDH1A1TSHRKDM4EHSD17B10MEN1
SCHEMBL23292188 0.66 PDE4A (0.42) ALDH1A1KDM4EPDE4APDE4CPDE4D
SCHEMBL17156594 0.65 TSHR (0.40) ALDH1A1TSHRKDM4EMEN1KMT2A
SCHEMBL249779 0.65 METAP2 (0.64) KDM4EPDE4APDE4CPDE4DSLC40A1
SCHEMBL16072722 0.64 KCNA3 (0.46) MAPTLMNAL3MBTL1MAPK1HTT
SCHEMBL6636842 0.64 PDE4A (0.43) KDM4EPDE4APDE4CPDE4DSLC40A1
SCHEMBL3515379 0.63 KDM4E (0.45) ALDH1A1TSHROPRM1OPRD1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2044068-A1 1-HYDROXY NAPHTHYRIDINE COMPOUNDS AS ANTI-HIV AGENTS Merck & Co., Inc. (US) 2009-04-08 EP disclosed
WO-2008010964-A1 1-HYDROXY NAPHTHYRIDINE COMPOUNDS AS ANTI-HIV AGENTS MERCK & CO., INC. (US) 2008-01-24 WO disclosed