SCHEMBL4490274

SCHEMBL4490274

NC(=O)Nc1c[nH]c2ccccc12

nearest known ligand 0.59

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
STING1 Q86WV6 13/20 0.59
ALDH1A1 P00352 1/20 0.58
ATM Q13315 1/20 0.58
GPR84 Q9NQS5 1/20 0.52
KDM4E B2RXH2 1/20 0.50
GAA P10253 1/20 0.50
STAT3 P40763 1/20 0.49
NR4A2 P43354 1/20 0.49
CREBBP Q92793 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14889338 0.88 STING1 (0.55) STING1ALDH1A1ATMGPR84GAA
SCHEMBL28736881 0.87 STING1 (0.74) STING1ALDH1A1ATMGPR84NR4A2
SCHEMBL384965 0.85 STING1 (0.63) STING1GPR84
SCHEMBL1596152 0.84 STING1 (0.61) STING1GPR84NR4A2CREBBP
SCHEMBL2884199 0.84 MAPK1 (0.63) STING1ALDH1A1ATMKDM4EGAA
SCHEMBL27522079 0.83 STING1 (0.54) STING1ALDH1A1ATMGPR84GAA
SCHEMBL5894412 0.82 STING1 (0.56) STING1ALDH1A1GPR84KDM4EGAA
SCHEMBL23167581 0.81 STING1 (0.58) STING1GPR84GAANR4A2CREBBP
SCHEMBL9347092 0.81 STING1 (0.58) STING1GPR84GAANR4A2CREBBP
SCHEMBL7543952 0.81 STING1 (0.55) STING1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 51 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115160209-B Indole group-containing compound and preparation method and application thereof 华南师范大学 2024-03-29 CN claimed
CN-115093361-B Novel indole acylhydrazone compound and preparation method and application thereof 华南师范大学 2024-02-13 CN claimed
WO-2023239903-A1 COMPOSITIONS AND METHODS FOR PREVENTING RETENTION OF PSMA-TARGETED THERAPY CASE WESTERN RESERVE UNIVERSITY (US) 2023-12-14 WO claimed
EP-4103278-A1 SMALL MOLECULE STING ANTAGONISTS Curadev Pharma Pvt. Ltd. (IN) 2022-12-21 EP claimed
CN-108101828-B 3-indolyl formamide compound and preparation method thereof 西华师范大学 2021-05-04 CN claimed
CN-119330982-A Azetidine compound and medical application thereof 中国科学院上海药物研究所 2025-01-21 CN disclosed
CN-117903038-A N-ethylcarbazole-3-indolyl formylhydrazone compound and preparation method thereof 佳木斯大学 2024-04-19 CN disclosed
CN-117777004-A Deuterated indolyl urea compound and medical application thereof 重庆中国药科大学创新研究院 2024-03-29 CN disclosed
CN-117777004-A Deuterated indolyl urea compound and medical application thereof 重庆中国药科大学创新研究院 2024-03-29 CN disclosed
CN-115160209-B Indole group-containing compound and preparation method and application thereof 华南师范大学 2024-03-29 CN disclosed
CN-117777004-A Deuterated indolyl urea compound and medical application thereof 重庆中国药科大学创新研究院 2024-03-29 CN disclosed
CN-117756698-A Urea compound and medical application thereof as STING inhibitor 中国药科大学 2024-03-26 CN disclosed
EP-0544819-B1 INDOLE DERIVATIVES WHICH INHIBIT LEUKOTRIENE BIOSYNTHESIS ABBOTT LAB (US) 1995-12-06 EP disclosed
US-5459150-A Treatment of allergies and inflammatory diseases ABBOTT LABORATORIES (US) 1995-10-17 US disclosed
EP-0544819-A4 INDOLE DERIVATIVES WHICH INHIBIT LEUKOTRIENE BIOSYNTHESIS 1993-10-20 EP disclosed
CN-1076197-A The preparation method of indole urea derivative BEECHAM GROUP PLC (GB) 1993-09-15 CN disclosed
CN-1076197-A The preparation method of indole urea derivative BEECHAM GROUP PLC (GB) 1993-09-15 CN disclosed
EP-0544819-A1 INDOLE DERIVATIVES WHICH INHIBIT LEUKOTRIENE BIOSYNTHESIS. ABBOTT LAB (US) 1993-06-09 EP disclosed
US-5095031-A Enzyme inhibitors, antiallergens, antiinflammatory ABBOTT LABORATORIES (US) 1992-03-10 US disclosed
WO-1992003132-A1 INDOLE DERIVATIVES WHICH INHIBIT LEUKOTRIENE BIOSYNTHESIS ABBOTT LABORATORIES (US) 1992-03-05 WO disclosed