SCHEMBL4495489

SCHEMBL4495489

CC1CCCCN1C(C(N)=O)c1c(C(=O)O)ccc2cc(OCCCN3CCCCC3)ccc12

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 8/20 0.48
MAOB P27338 7/20 0.45
MET P08581 1/20 0.43
HRH1 P35367 1/20 0.42
DHODH Q02127 1/20 0.41
POLB P06746 1/20 0.41
MAPT P10636 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4509193 0.79 MAOB (0.48) HRH3MAOBPOLBMAPTKDM4E
SCHEMBL4502216 0.76 HRH3 (0.45) HRH3MAOBMETKDM4EALDH1A1
SCHEMBL4501682 0.74 HRH3 (0.48) HRH3MAOBMETHRH1POLB
SCHEMBL4501879 0.73 HRH3 (0.52) HRH3MAOBMET
SCHEMBL4505175 0.72 HRH3 (0.50) HRH3MAOBPOLBMAPTKDM4E
SCHEMBL4501323 0.72 HRH3 (0.73) HRH3MAOBKDM4E
SCHEMBL4505136 0.72 HRH3 (0.48) HRH3MAOBMET
SCHEMBL4490641 0.71 HRH3 (0.49) HRH3MAOBHRH1
SCHEMBL4503090 0.70 HRH3 (0.73) HRH3MAOBPOLBMAPTKDM4E
SCHEMBL4506214 0.69 HRH3 (0.55) HRH3MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7608617-B2 Naphthaline derivatives as H3 inverse agonists HOFFMANN-LA ROCHE INC. (US) 2009-10-27 US disclosed