SCHEMBL4502216

SCHEMBL4502216

NC(=O)C(c1cccs1)c1c(C(=O)O)ccc2cc(OCCCN3CCCCC3)ccc12

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 12/20 0.45
MAOB P27338 4/20 0.43
KCNH2 Q12809 2/20 0.43
MET P08581 1/20 0.42
KDM4E B2RXH2 3/20 0.41
ALDH1A1 P00352 3/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4509193 0.78 MAOB (0.48) HRH3MAOBKDM4EALDH1A1KMT2A
SCHEMBL4495489 0.76 HRH3 (0.48) HRH3MAOBMETKDM4EALDH1A1
SCHEMBL4505175 0.71 HRH3 (0.50) HRH3MAOBKCNH2KDM4EALDH1A1
SCHEMBL4501682 0.69 HRH3 (0.48) HRH3MAOBMETKDM4EALDH1A1
SCHEMBL4488748 0.69 HRH3 (0.77) HRH3MAOBKDM4EALDH1A1SMN1; SMN2
SCHEMBL3296967 0.69 MAOB (0.79) MAOBMETKDM4EALDH1A1SMN1; SMN2
SCHEMBL4498291 0.69 NPC1 (0.54) HRH3MAOBMETKDM4EALDH1A1
Hydrochloric Acid SCHEMBL7628740 0.69 GCGR (0.60) HRH3KDM4E
SCHEMBL5107040 0.68 MAOB (0.62) HRH3MAOBMETKDM4EALDH1A1
SCHEMBL3131412 0.68 MAOB (0.59) HRH3MAOBKDM4EALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7608617-B2 Naphthaline derivatives as H3 inverse agonists HOFFMANN-LA ROCHE INC. (US) 2009-10-27 US disclosed