SCHEMBL4495537

SCHEMBL4495537

CC(C)c1c(C#Cc2ccccn2)[nH]c(C=O)c1C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 1/20 0.39
FFAR1 O14842 1/20 0.36
GRM5 P41594 4/20 0.35
HAO1 Q9UJM8 2/20 0.35
CLK2 P49760 1/20 0.35
KDR P35968 1/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4489156 0.83 FFAR1 (0.37) FFAR1GRM5
SCHEMBL4482502 0.75 FLT4 (0.30)
SCHEMBL4490782 0.73 GRM5 (0.40) ERN1FFAR1GRM5KDRPTGDR2
SCHEMBL4494939 0.72
SCHEMBL4490395 0.72
SCHEMBL4505401 0.70 ALDH1A1 (0.30)
SCHEMBL4491011 0.70 SMN1; SMN2 (0.44)
SCHEMBL4491755 0.70 TRPV1 (0.36)
SCHEMBL4497337 0.69
SCHEMBL4486266 0.68 ALDH1A1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7504429-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2009-03-17 US claimed