SCHEMBL4497491

SCHEMBL4497491

O=C(O)c1ccc2[nH]c(NC(Cc3cccc4ccccc34)C3CCNCC3)nc2c1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.38
ABL1 P00519 2/20 0.38
CSNK2A1 P68400 1/20 0.37
CTNNB1 P35222 1/20 0.36
SENP2 Q9HC62 1/20 0.35
SENP1 Q9P0U3 1/20 0.35
SLC6A4 P31645 1/20 0.35
ACP1 P24666 2/20 0.34
MEN1 O00255 1/20 0.34
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
PIN1 Q13526 1/20 0.34
KDR P35968 1/20 0.33
ULK1 O75385 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4509585 0.91 SMN1; SMN2 (0.37) ABL1ACP1MEN1MAPTKMT2A
SCHEMBL4496677 0.86 SLC6A4 (0.34) SLC6A4MEN1MAPTKMT2ATDP1
SCHEMBL4494905 0.85 MAPK10 (0.40) SLC6A4ACP1
SCHEMBL4507517 0.83 ADRB2 (0.34) SLC6A4TDP1
SCHEMBL4503597 0.80 HDAC6 (0.43) AKR1C3ABL1CSNK2A1
SCHEMBL4493813 0.74 ALDH1A1 (0.37) SLC6A4MEN1MAPTKMT2A
SCHEMBL4497481 0.72 SMN1; SMN2 (0.44) SLC6A4
SCHEMBL4514607 0.72 KMT2A (0.38) MEN1MAPTKMT2A
SCHEMBL4502218 0.71 MEN1 (0.38) SLC6A4MEN1KMT2A
SCHEMBL4491405 0.66 KCNN1 (0.41) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7517875-B2 Piperidine derivatives having CCR3 antagonism TEIJIN LIMITED (JP) 2009-04-14 US disclosed
US-20070032525-A1 Piperidine derivatives having ccr3 antagonism TEIJIN LIMITED, A JAPANESE BODY CORPORATE (JP) 2007-02-08 US disclosed
EP-1502916-A1 PIPERIDINE DERIVATIVES HAVING CCR3 ANTAGONISM TEIJIN LIMITED (JP) 2005-02-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070032525-A1 Piperidine derivatives having ccr3 antagonism CCR3, CCR1, CCR4 AKR1C3 380/4885ABL1 3759/4885CSNK2A1 2738/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.