SCHEMBL4498539

SCHEMBL4498539

Cc1ccc(Cc2cccc(F)c2)o1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.50
IDH1 O75874 1/20 0.42
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41
IDO1 P14902 2/20 0.41
AGXT P21549 2/20 0.41
DAO P14920 1/20 0.40
ACHE P22303 1/20 0.39
POLB P06746 2/20 0.39
MEN1 O00255 1/20 0.39
CHRM2 P08172 1/20 0.39
CHRM4 P08173 1/20 0.39
CHRM5 P08912 1/20 0.39
CHRM1 P11229 1/20 0.39
CYP2C9 P11712 1/20 0.39
CHRM3 P20309 1/20 0.39
KMT2A Q03164 1/20 0.39
TP53 P04637 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
ADORA2A P29274 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4505633 0.82 MAPT (0.46) TAAR1IDO1DAOACHEPOLB
SCHEMBL4485406 0.81 TAAR1 (0.51) TAAR1MAOAMAOBIDO1AGXT
SCHEMBL25128958 0.79 MAPT (0.44) MAOAMAOBACHEPOLBMEN1
SCHEMBL1680634 0.79 TAAR1 (0.50) TAAR1MAOBIDO1AGXTDAO
SCHEMBL4492592 0.78 POLB (0.45) TAAR1MAOAMAOBPOLBMEN1
SCHEMBL4674508 0.78 ALDH1A1 (0.46) IDH1MAOAMAOBPOLBMEN1
SCHEMBL3180066 0.77 CHRM2 (0.47) TAAR1POLBMEN1CHRM2CHRM4
SCHEMBL4498868 0.77 CHRM2 (0.53) TAAR1IDH1MAOBIDO1AGXT
Water SCHEMBL9667780 0.76 CHRM2 (0.45) TAAR1POLBMEN1CHRM2CHRM4
SCHEMBL1680877 0.76 ALDH1A1 (0.46) TAAR1IDH1MAOAMAOBIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7576198-B1 Integrase inhibitors containing aromatic heterocycle derivatives SHIONOGI & CO., LTD. (JP) 2009-08-18 US disclosed
EP-1219607-A1 INTEGRASE INHIBITORS CONTAINING AROMATIC HETEROCYCLE DERIVATIVES SHIONOGI & CO., LTD. (JP) 2002-07-03 EP disclosed