SCHEMBL4499672

SCHEMBL4499672

Cc1cc(Br)ccc1-c1nnc(-c2cccc(OC(C)(C)C#N)c2)s1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.36
S1PR1 P21453 9/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
NOTUM Q6P988 1/20 0.35
HDAC1 Q13547 5/20 0.35
HDAC2 Q92769 5/20 0.35
HDAC8 Q9BY41 2/20 0.34
HDAC6 Q9UBN7 2/20 0.34
PIM1 P11309 1/20 0.34
PIM3 Q86V86 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6434492 0.71 MEN1 (0.39) KDM4ESMN1; SMN2
SCHEMBL4366155 0.68 S1PR1 (0.66) S1PR1
SCHEMBL4499678 0.68 S1PR1 (0.43) S1PR1
SCHEMBL4499675 0.67 S1PR1 (0.44) S1PR1
SCHEMBL4373320 0.66 S1PR1 (0.46) S1PR1
SCHEMBL4561969 0.64 S1PR1 (0.60) S1PR1
SCHEMBL6588477 0.64 SMN1; SMN2 (0.52) SMN1; SMN2HDAC8
SCHEMBL4369991 0.64 S1PR1 (0.47) S1PR1
SCHEMBL1180747 0.63 RAB9A (0.59) KDM4ESMN1; SMN2NOTUMPIM1PIM3
SCHEMBL22347377 0.62 ALDH1A1 (0.41) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7605171-B2 (3,4-disubstituted)propanoic carboxylates as S1P (Edg) receptor agonists MERCK & CO., INC. (US) 2009-10-20 US disclosed
US-20080249093-A1 (3,4-Disubstituted)Propanoic Carboxylates as Sip (Edg) Receptor Agonists MERCK & CO., INC. (US) 2008-10-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080249093-A1 (3,4-Disubstituted)Propanoic Carboxylates as Sip (Edg) Receptor Agonists S1PR1, S1PR3, S1PR5 KDM4E 2051/4885S1PR1 1/4885SMN1; SMN2 2376/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.