SCHEMBL4500503

SCHEMBL4500503

Cc1ccc(-c2ccc3c(NC(=O)c4cccc(F)c4)n[nH]c3c2)cc1C

nearest known ligand 0.58

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
FGFR2 P21802 3/20 0.58
FGFR3 P22607 3/20 0.58
FGFR1 P11362 2/20 0.58
GSK3B P49841 3/20 0.58
GSK3A P49840 1/20 0.58
HDAC6 Q9UBN7 14/20 0.55
FGFR4 P22455 1/20 0.52
CYP1A2 P05177 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4489751 0.89 HDAC6 (0.61) FGFR2FGFR3FGFR1GSK3BGSK3A
SCHEMBL4485646 0.89 HDAC6 (0.70) FGFR2FGFR3FGFR1GSK3BGSK3A
SCHEMBL4480304 0.89 HDAC6 (0.59) FGFR2FGFR3FGFR1GSK3BGSK3A
SCHEMBL4483456 0.88 HDAC6 (0.61) FGFR2FGFR3FGFR1GSK3BGSK3A
SCHEMBL4498043 0.87 GSK3B (0.61) FGFR2FGFR3FGFR1GSK3BGSK3A
SCHEMBL4491728 0.87 FGFR1 (0.61) FGFR2FGFR3FGFR1GSK3BGSK3A
SCHEMBL4489919 0.87 HDAC6 (0.54) FGFR2FGFR3FGFR1GSK3BGSK3A
SCHEMBL4488600 0.86 HDAC6 (0.61) FGFR2FGFR3FGFR1GSK3BHDAC6
SCHEMBL4492924 0.85 HDAC6 (0.70) FGFR2FGFR3FGFR1GSK3BGSK3A
SCHEMBL4558929 0.85 HDAC6 (0.74) FGFR2FGFR3FGFR1GSK3BGSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7632854-B2 Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them PFIZER ITALIA S.R.L. (IT) 2009-12-15 US claimed