SCHEMBL4501039

SCHEMBL4501039

Cc1cc(CCl)cc(Cl)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.44
HTT P42858 2/20 0.44
LMNA P02545 2/20 0.39
ALDH1A1 P00352 2/20 0.36
MAPK1 P28482 1/20 0.36
KDM4E B2RXH2 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
HIF1A Q16665 1/20 0.36
KMT2A Q03164 3/20 0.35
RECQL P46063 1/20 0.34
MEN1 O00255 1/20 0.34
ADORA2A P29274 2/20 0.33
ADORA1 P30542 2/20 0.33
GRM5 P41594 1/20 0.33
NPSR1 Q6W5P4 1/20 0.32
POLB P06746 1/20 0.32
APOBEC3G Q9HC16 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
ADORA2B P29275 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29560985 1.00 SMN1; SMN2 (0.44) SMN1; SMN2HTTLMNAALDH1A1MAPK1
SCHEMBL1314802 0.87 HTT (0.43) SMN1; SMN2HTTLMNAKMT2AMEN1
SCHEMBL501235 0.86 RECQL (0.45) SMN1; SMN2HTTLMNAALDH1A1MAPK1
Hydrochloric Acid SCHEMBL502252 0.85 HTT (0.42) SMN1; SMN2HTTLMNAALDH1A1MAPK1
SCHEMBL9608992 0.84 NPC1 (0.39) SMN1; SMN2HTTLMNAALDH1A1MAPK1
SCHEMBL29714427 0.82 LOX (0.45) SMN1; SMN2HTTLMNAALDH1A1MAPK1
SCHEMBL19755849 0.82 LOX (0.45) SMN1; SMN2HTTLMNAALDH1A1MAPK1
SCHEMBL6931382 0.82 HTT (0.37) SMN1; SMN2HTTLMNAALDH1A1MAPK1
SCHEMBL5898063 0.82 HTT (0.41) SMN1; SMN2HTTLMNAALDH1A1MAPK1
SCHEMBL190086 0.82 RECQL (0.41) SMN1; SMN2HTTALDH1A1KDM4ECYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 76 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3334721-B1 CGRP RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2021-04-28 EP disclosed
EP-3341370-B1 CGRP RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2021-04-28 EP disclosed
CN-107922385-B CGRP receptor antagonists 伊莱利利公司 2020-09-08 CN disclosed
CN-107922406-B CGRP receptor antagonists 伊兰科美国公司 2020-04-03 CN disclosed
EP-3341370-A1 CGRP RECEPTOR ANTAGONISTS Eli Lilly and Company (US) 2018-07-04 EP disclosed
CN-105283453-B N- (pyridin-2-yl) pyrimidin-4-amine derivatives containing sulfone group 拜耳药业股份公司 2018-06-22 CN disclosed
EP-3334721-A1 CGRP RECEPTOR ANTAGONISTS Eli Lilly and Company (US) 2018-06-20 EP disclosed
CN-107922385-A Cgrp receptor antagonists 伊莱利利公司 2018-04-17 CN disclosed
CN-107922406-A CGRP receptor antagonist 伊莱利利公司 2018-04-17 CN disclosed
US-9877954-B2 5-fluoro-N-(pyridin-2-yl)pyridin-2-amine derivatives containing a sulfoximine group BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2018-01-30 US disclosed
US-5298507-A Insecticides NIHON BAYER AGROCHEM K.K. (JP) 1994-03-29 US disclosed
US-5204360-A Insecticides NIHON BAYER AGROCHEM K.K. (JP) 1993-04-20 US disclosed
US-5001138-A Insecticides NIHON TOKUSHU NOYAKU SEIZO, K.K. (JP) 1991-03-19 US disclosed
US-4845106-A INSECTICIDES NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1989-07-04 US disclosed
US-4812571-A NITROMETHYLENE COMPOUNDS NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1989-03-14 US disclosed
US-4774247-A Nitromethylene derivative insecticides NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1988-09-27 US disclosed
US-4742060-A 2-(NITROIMINO)- OR 2-(NITROMETHYLENE)-IMIDAZOLIDINES AS INSECTICIDES NIHON TOKUSHU NOYAKU SEIZO K. K. (JP) 1988-05-03 US disclosed
US-4678795-A 1-pyridylmethyl-2-nitromethylene-1,3-diazacycloalkane insecticides NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1987-07-07 US disclosed
EP-0192060-A1 Heterocyclic compounds NIHON BAYER AGROCHEM K.K. (JP) 1986-08-27 EP disclosed
EP-0163855-A1 Nitromethylene derivatives, intermediates, and process for their preparation as insecticides NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1985-12-11 EP disclosed