SCHEMBL4522246

SCHEMBL4522246

O=C(C=Cc1cccc(S(=O)(=O)N2CCN(Cc3ccccc3)CC2I)c1)NO

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 18/20 0.54
HDAC3 O15379 17/20 0.54
HDAC4 P56524 17/20 0.54
HDAC7 Q8WUI4 17/20 0.54
HDAC2 Q92769 17/20 0.54
HDAC8 Q9BY41 17/20 0.54
HDAC6 Q9UBN7 17/20 0.54
HDAC9 Q9UKV0 17/20 0.54
HDAC5 Q9UQL6 17/20 0.54
HDAC10 Q969S8 16/20 0.54
HDAC11 Q96DB2 16/20 0.54
KCNH2 Q12809 1/20 0.50
BCHE P06276 2/20 0.48
ACHE P22303 2/20 0.48
BRD4 O60885 1/20 0.48
ESR1 P03372 1/20 0.48
PTGS1 P23219 1/20 0.48
PDE4A P27815 1/20 0.48
PIK3CA P42336 1/20 0.48
HTR6 P50406 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6493407 0.88 HDAC1 (0.52) HDAC1HDAC3HDAC4HDAC7HDAC2
SCHEMBL1376403 0.84 HDAC1 (0.73) HDAC1HDAC3HDAC4HDAC7HDAC2
SCHEMBL1376399 0.84 HDAC1 (0.73) HDAC1HDAC3HDAC4HDAC7HDAC2
SCHEMBL4508022 0.79 HDAC1 (0.72) HDAC1HDAC3HDAC4HDAC7HDAC2
SCHEMBL12152501 0.76 HDAC1 (0.70) HDAC1HDAC3HDAC4HDAC7HDAC2
SCHEMBL1376425 0.74 HDAC1 (0.72) HDAC1HDAC3HDAC4HDAC7HDAC2
SCHEMBL1376427 0.74 HDAC1 (0.72) HDAC1HDAC3HDAC4HDAC7HDAC2
SCHEMBL1486911 0.73 HDAC1 (0.64) HDAC1HDAC3HDAC4HDAC7HDAC2
SCHEMBL1486915 0.73 HDAC1 (0.64) HDAC1HDAC3HDAC4HDAC7HDAC2
SCHEMBL12152302 0.73 ALDH1A1 (0.61) HDAC1HDAC3HDAC4HDAC7HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7629343-B2 Carbamic acid compounds comprising a piperazine linkage as HDAC inhibitors TOPOTARGET UK LIMITED (GB) 2009-12-08 US disclosed
EP-1492534-B1 CARBAMIC ACID COMPOUNDS COMPRISING A PIPERAZINE LINKAGE AS HDAC INHIBITORS TOPOTARGET UK LTD (GB) 2008-06-25 EP disclosed