SCHEMBL4524967

SCHEMBL4524967

O=C(ON1C(=O)CCC1=O)C(Br)CBr

nearest known ligand 0.37

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.37
TSHR P16473 1/20 0.37
MGLL Q99685 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18885710 0.82 MGLL (0.36) MGLL
SCHEMBL7092660 0.80 MGLL (0.35) MGLL
SCHEMBL1906467 0.78 MGLL (0.34) MGLL
SCHEMBL4867939 0.78 ZDHHC7 (0.47) ALDH1A1TSHR
SCHEMBL4422537 0.76 ALDH1A1 (0.31) ALDH1A1TSHR
SCHEMBL1275225 0.76 CYP2C19 (0.41) ALDH1A1MGLL
SCHEMBL20404645 0.75 MGLL (0.36) MGLL
SCHEMBL111364 0.75 MGLL (0.36) MGLL
SCHEMBL37884 0.75 MGLL (0.36) MGLL
SCHEMBL2573222 0.75 MGLL (0.36) MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 28 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113301928-B Biological scaffolds and methods for making same 黄玲惠 2022-12-02 CN claimed
EP-0977588-B1 COUPLING OF UNMODIFIED PROTEINS TO HALOACYL OR DIHALOACYL DERIVATIZED POLYSACCHARIDES FOR THE PREPARATION OF PROTEIN-POLYSACCHARIDE VACCINES JACKSON H M FOUND MILITARY MED (US) 2004-10-06 EP claimed
US-6087328-A FUNCTIONALIZING A POLYSACCHARIDE WITH ONE OR MORE PENDANT HALOACYL GROUPS, THEN THE FUNCTIONALIZED GROUP IS REACTED WITH PROTEIN OR PEPTIDE TO FORM A COVALENTLY LINKED CONJUGATE, USEFUL AS A VACCINE AGAINST BACTERIA, FUNGI OR VIRUSES HENRY M. JACKSON FOUNDATION FOR THE ADVANCEMENT OF MILITARY MEDICINE (US) 2000-07-11 US claimed
EP-0977588-A2 COUPLING OF UNMODIFIED PROTEINS TO HALOACYL OR DIHALOACYL DERIVATIZED POLYSACCHARIDES FOR THE PREPARATION OF PROTEIN-POLYSACCHARIDE VACCINES HENRY M. JACKSON FOUNDATION FOR THE ADVANCEMENT OF MILITARY MEDICINE (US) 2000-02-09 EP claimed
WO-1998047530-A2 COUPLING OF UNMODIFIED PROTEINS TO HALOACYL OR DIHALOACYL DERIVATIZED POLYSACCHARIDES FOR THE PREPARATION OF PROTEIN-POLYSACCHARIDE VACCINES HENRY M. JACKSON FOUNDATION FOR THE ADVANCEMENT OF MILITARY MEDICINE (US) 1998-10-29 WO claimed
CN-115869468-B Biological scaffold and method for preparing the same 黄玲惠 2025-02-14 CN disclosed
CN-115869468-A Biological scaffolds and methods for making same 黄玲惠 2023-03-31 CN disclosed
CN-113301928-B Biological scaffolds and methods for making same 黄玲惠 2022-12-02 CN disclosed
CN-105131104-B The reconstruct and sugar conjugation of peptide 诺和诺德公司 2018-11-16 CN disclosed
US-20090305264-A1 COOPERATIVE PROBES AND METHODS OF USING THEM FLUIDIGM CORPORATION 2009-12-10 US disclosed
EP-2004861-A2 COOPERATIVE PROBES AND METHODS OF USING THEM Arcxis Biotechnologies, Inc. (US) 2008-12-24 EP disclosed
EP-1893741-A1 CELL-BASED MICROARRAYS, AND METHODS FOR THEIR PREPARATION AND USE Beckman Coulter, Inc. (US) 2008-03-05 EP disclosed
EP-0977588-A2 COUPLING OF UNMODIFIED PROTEINS TO HALOACYL OR DIHALOACYL DERIVATIZED POLYSACCHARIDES FOR THE PREPARATION OF PROTEIN-POLYSACCHARIDE VACCINES HENRY M. JACKSON FOUNDATION FOR THE ADVANCEMENT OF MILITARY MEDICINE (US) 2000-02-09 EP disclosed
EP-0977588-A2 COUPLING OF UNMODIFIED PROTEINS TO HALOACYL OR DIHALOACYL DERIVATIZED POLYSACCHARIDES FOR THE PREPARATION OF PROTEIN-POLYSACCHARIDE VACCINES HENRY M. JACKSON FOUNDATION FOR THE ADVANCEMENT OF MILITARY MEDICINE (US) 2000-02-09 EP disclosed
WO-1998047530-A3 COUPLING OF UNMODIFIED PROTEINS TO HALOACYL OR DIHALOACYL DERIVATIZED POLYSACCHARIDES FOR THE PREPARATION OF PROTEIN-POLYSACCHARIDE VACCINES LEES ANDREW C (US) 1999-01-28 WO disclosed
WO-1998047530-A2 COUPLING OF UNMODIFIED PROTEINS TO HALOACYL OR DIHALOACYL DERIVATIZED POLYSACCHARIDES FOR THE PREPARATION OF PROTEIN-POLYSACCHARIDE VACCINES HENRY M. JACKSON FOUNDATION FOR THE ADVANCEMENT OF MILITARY MEDICINE (US) 1998-10-29 WO disclosed
WO-1998047530-A2 COUPLING OF UNMODIFIED PROTEINS TO HALOACYL OR DIHALOACYL DERIVATIZED POLYSACCHARIDES FOR THE PREPARATION OF PROTEIN-POLYSACCHARIDE VACCINES HENRY M. JACKSON FOUNDATION FOR THE ADVANCEMENT OF MILITARY MEDICINE (US) 1998-10-29 WO disclosed
US-5648213-A IMMUNOASSAY BECKMAN INSTRUMENTS, INC. (US) 1997-07-15 US disclosed
EP-0779934-A1 COMPOSITIONS AND METHODS FOR USE IN DETECTION OF ANALYTES BECKMAN INSTRUMENTS, INC. (US) 1997-06-25 EP disclosed
WO-1996006948-A1 COMPOSITIONS AND METHODS FOR USE IN DETECTION OF ANALYTES BECKMAN INSTRUMENTS, INC. (US) 1996-03-07 WO disclosed