SCHEMBL453284

SCHEMBL453284

O=C(O)c1ccccc1/N=N/c1ccc(O)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDE P14735 1/20 1.00
KMT2A Q03164 9/20 0.68
MEN1 O00255 8/20 0.68
MAPT P10636 5/20 0.68
MYC P01106 1/20 0.67
NPC1 O15118 1/20 0.59
NPSR1 Q6W5P4 3/20 0.58
GAA P10253 3/20 0.58
L3MBTL1 Q9Y468 2/20 0.58
TDP1 Q9NUW8 3/20 0.56
THRB P10828 2/20 0.56
PSMD14 O00487 1/20 0.56
HSP90AA1 P07900 1/20 0.56
MMP2 P08253 1/20 0.56
MAPK1 P28482 1/20 0.56
POLB P06746 2/20 0.50
TRPA1 O75762 1/20 0.48
CCNE2 O96020 1/20 0.47
CCNE1 P24864 1/20 0.47
CDK2 P24941 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL453285 1.00 IDE (1.00) IDEKMT2AMEN1MAPTMYC
SCHEMBL29401042 1.00 IDE (1.00) IDEKMT2AMEN1MAPTMYC
SCHEMBL12100493 1.00 IDE (1.00) IDEKMT2AMEN1MAPTMYC
SCHEMBL30884072 0.89 IDE (0.79) IDEKMT2AMEN1MAPTMYC
SCHEMBL28903951 0.89 IDE (0.79) IDEKMT2AMEN1MAPTMYC
SCHEMBL2481541 0.89 IDE (0.79) IDEKMT2AMEN1MAPTMYC
SCHEMBL169230 0.89 IDE (0.79) IDEKMT2AMEN1MAPTMYC
Phenol SCHEMBL7057355 0.89 IDE (0.79) IDEKMT2AMEN1MAPTMYC
SCHEMBL28229539 0.87 IDE (0.77) IDEKMT2AMEN1MAPTMYC
SCHEMBL28229538 0.87 IDE (0.77) IDEKMT2AMEN1MAPTMYC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 982 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4661890-A1 PTP1B/TC-PTP DUAL INHIBITORS AND PROTEIN DEGRADERS Purdue Research Foundation (US) 2025-12-17 EP claimed
US-20250027947-A1 KITS, MICROFLUIDICS DEVICES, AND METHODS FOR PERFORMING BIOTIN ASSAYS SIEMENS HEALTHCARE DIAGNOSTICS INC. (US) 2025-01-23 US claimed
US-12168801-B1 Hybrid/capture probe designs for full-length cDNA 10X GENOMICS, INC. (US) 2024-12-17 US claimed
US-20240399022-A1 COMPOSITIONS AND METHODS FOR MACROPHAGE CONVERSION UNIV DREXEL (US) 2024-12-05 US claimed
EP-3830556-B1 KITS, MICROFLUIDICS DEVICES, AND METHODS FOR PERFORMING BIOTIN ASSAYS SIEMENS HEALTHCARE DIAGNOSTICS INC (US) 2024-11-13 EP claimed
US-12140596-B2 Kits, microfluidics devices, and methods for performing biotin assays SIEMENS HEALTHCARE DIAGNOSTICS INC. (US) 2024-11-12 US claimed
US-12077819-B2 Compositions and processes for improved mass spectrometry analysis AGENA BIOSCIENCE, INC. (US) 2024-09-03 US claimed
WO-2024167565-A1 PTP1B/TC-PTP DUAL INHIBITORS AND PROTEIN DEGRADERS PURDUE RESEARCH FOUNDATION (US) 2024-08-15 WO claimed
US-20240096612-A1 METHOD FOR MASS SPECTROMETRY OF ORGANIC SYNTHETIC COMPOUND SHIMADZU CORPORATION (JP) 2024-03-21 US claimed
CN-117720438-A Preparation method of multifunctional perfluorinated acrylate monomer 江苏三木化工股份有限公司 2024-03-19 CN claimed
WO-2004023147-A2 MALDI-MATRIX N.V. NUTRICIA (NL) 2004-03-18 WO claimed
US-6632929-B1 Conjugate with 4'-hydroxyazobenzene-2-carboxylic acid derivative; change from red to yellow upon binding biotin YEDA RESEARCH AND DEVELOPMENT CO. LTD (IL) 2003-10-14 US claimed
WO-2003050517-A1 OPTICALLY TRANSPARENT SUBSTRATE FOR A MALDI MEASURING SYSTEM AND THE USE THEREOF ZEPTOSENS AG (CH) 2003-06-19 WO claimed
US-6110641-A Radiation sensitive composition containing novel dye SHIPLEY COMPANY, L.L.C. (US) 2000-08-29 US claimed
WO-2000027813-A1 AZOBENZENE DERIVATIVES AS LABELING AGENTS AND INTERMEDIATES THEREOF YEDA RESEARCH AND DEVELOPMENT CO. LTD. (IL) 2000-05-18 WO claimed
WO-2000027814-A1 AVIDIN DERIVATIVES AND USES THEREOF YEDA RESEARCH AND DEVELOPMENT CO. LTD. (IL) 2000-05-18 WO claimed
US-5770272-A Matrix-bearing targets for maldi mass spectrometry and methods of production thereof MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 1998-06-23 US claimed
US-5763191-A BINDING MATRIX BOEHRINGER MANNHEIM GMBH (DE) 1998-06-09 US claimed
WO-1996033797-A1 MATRIX-BEARING TARGETS FOR MALDI MASS SPECTROMETRY AND METHODS OF PRODUCTION THEREOF MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 1996-10-31 WO claimed
EP-0571087-A1 Cleavable phosphoramidites ROHM AND HAAS COMPANY (US) 1993-11-24 EP claimed