SCHEMBL4535793

SCHEMBL4535793

O=Cc1[nH]nnc1Cc1ccccc1F

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.48
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 1/20 0.38
DAO P14920 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
HCAR3 P49019 1/20 0.35
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
AKR1B1 P15121 1/20 0.34
P2RX7 Q99572 1/20 0.34
TAAR1 Q96RJ0 2/20 0.33
GUCY1A1 Q02108 1/20 0.33
GUCY1B1 Q02153 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20578752 0.71 AR (0.52) ARALDH1A1KDM4EDAOMEN1
SCHEMBL5776720 0.70 AR (0.48) ARALDH1A1KDM4EDAOMEN1
SCHEMBL18965577 0.68 ADRA1D (0.45) AKR1B1
SCHEMBL16401681 0.67 AR (0.41) ARALDH1A1KDM4EDAOHCAR3
SCHEMBL16781994 0.66 ALDH1A1 (0.47) ARALDH1A1DAOMEN1KMT2A
SCHEMBL28804739 0.66 ALDH1A1 (0.41) ARALDH1A1KDM4EDAOHTT
SCHEMBL3301625 0.65 TAAR1 (0.59) ARALDH1A1KDM4EDAOTAAR1
SCHEMBL12955359 0.65 AR (1.00) ARHTT
SCHEMBL3581160 0.64 AR (0.68) ARALDH1A1KDM4E
SCHEMBL12468870 0.62 IDO1 (0.40) ARALDH1A1KDM4EDAOMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2638029-A1 TRIAZOLE DERIVATIVES AND THEIR USE FOR NEUROLOGICAL DISORDERS F.HOFFMANN-LA ROCHE AG (CH) 2013-09-18 EP disclosed
WO-2012062687-A1 TRIAZOLE DERIVATIVES AND THEIR USE FOR NEUROLOGICAL DISORDERS F. HOFFMANN-LA ROCHE AG (CH) 2012-05-18 WO disclosed