SCHEMBL4535957

SCHEMBL4535957

O=C(CC1CCNCC1)NC12CC3CC(CC(C3)C1)C2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 7/20 1.00
EPHX2 P34913 6/20 0.64
CACNA1H O95180 1/20 0.49
HDAC3 O15379 1/20 0.47
HDAC4 P56524 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC7 Q8WUI4 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC10 Q969S8 1/20 0.47
HDAC11 Q96DB2 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
HDAC9 Q9UKV0 1/20 0.47
HDAC5 Q9UQL6 1/20 0.47
ATM Q13315 1/20 0.46
ALDH1A1 P00352 3/20 0.45
MEN1 O00255 1/20 0.45
MAPT P10636 1/20 0.45
KMT2A Q03164 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4537511 0.91 EPHX1 (0.84) EPHX1EPHX2CACNA1HHDAC3HDAC4
SCHEMBL19798447 0.83 EPHX1 (0.71) EPHX1EPHX2CACNA1HHDAC3HDAC4
SCHEMBL4542363 0.82 EPHX1 (1.00) EPHX1EPHX2CACNA1HHDAC3HDAC4
SCHEMBL30618915 0.81 EPHX1 (0.68) EPHX1EPHX2HDAC3HDAC1HDAC8
SCHEMBL8925408 0.78 EPHX2 (1.00) EPHX1EPHX2
Hydrochloric Acid SCHEMBL18686528 0.78 EPHX1 (0.64) EPHX1EPHX2CACNA1HHDAC3HDAC4
Hydrochloric Acid SCHEMBL18686624 0.78 EPHX1 (0.64) EPHX1EPHX2CACNA1HHDAC3HDAC4
SCHEMBL4228257 0.78 EPHX1 (0.64) EPHX1EPHX2HDAC3HDAC4HDAC1
Hydrochloric Acid SCHEMBL18686525 0.78 EPHX1 (0.64) EPHX1EPHX2CACNA1HHDAC3HDAC4
SCHEMBL19173156 0.78 EPHX1 (0.62) EPHX1EPHX2ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed