SCHEMBL4538554

SCHEMBL4538554

CON=Cc1cccc2[nH]cnc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.43
PARP1 P09874 1/20 0.40
RET P07949 1/20 0.36
ADRA1D P25100 1/20 0.35
ADRA1A P35348 1/20 0.35
ADRA1B P35368 1/20 0.35
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
MAPT P10636 2/20 0.35
KDM4E B2RXH2 1/20 0.35
KMT2A Q03164 1/20 0.35
MMP12 P39900 1/20 0.35
DRD4 P21917 3/20 0.35
DRD3 P35462 3/20 0.35
DRD2 P14416 2/20 0.35
ABL1 P00519 1/20 0.34
RAD52 P43351 1/20 0.34
RIN1 Q13671 1/20 0.34
HTR2A P28223 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4537910 0.79 PARP1 (0.46) BRD4PARP1MAPTKDM4EKMT2A
SCHEMBL8051296 0.76 PARP1 (0.46) BRD4PARP1RETMAPTKMT2A
SCHEMBL16502119 0.73 PARP1 (0.46) BRD4PARP1RETMAPTKMT2A
SCHEMBL534330 0.73 PARP1 (0.50) BRD4PARP1RETMAPTKMT2A
Hydrochloric Acid SCHEMBL28064657 0.71 PARP1 (0.49) BRD4PARP1RETMAPTKMT2A
SCHEMBL3578437 0.71 TUBB4A (0.43) PARP1
SCHEMBL13343596 0.71 TUBB4A (0.43) PARP1
SCHEMBL23676438 0.71 HSD17B10 (0.39) PARP1ADRA1DADRA1AADRA1BADRA2A
SCHEMBL10140 0.69 BRD4 (0.60) BRD4PARP1RETKMT2AMMP12
SCHEMBL536589 0.67 PARP1 (0.64) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2638007-A2 DRUG DERIVATIVES Redx Pharma Limited (GB) 2013-09-18 EP disclosed
WO-2012063085-A2 DRUG DERIVATIVES REDX PHARMA LIMITED (GB) 2012-05-18 WO disclosed