SCHEMBL4539301

SCHEMBL4539301

CS(=O)(=O)c1ccc(N2CCN(Cc3ccccc3)CC2)cc1

nearest known ligand 0.73

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.73
DRD4 P21917 3/20 0.66
LMNA P02545 1/20 0.64
CCR2 P41597 2/20 0.56
HTR2A P28223 1/20 0.54
HTR2C P28335 1/20 0.54
HTR2B P41595 1/20 0.54
L3MBTL1 Q9Y468 1/20 0.54
TSHR P16473 1/20 0.53
LSS P48449 1/20 0.53
SIGMAR1 Q99720 1/20 0.53
HSP90AA1 P07900 1/20 0.52
HSP90AB1 P08238 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22516947 0.87 DRD2 (0.56) DRD2DRD4LMNALSSHSP90AA1
SCHEMBL6442002 0.85 DRD4 (0.66) DRD2DRD4HTR2AHTR2CHTR2B
SCHEMBL8781020 0.82 DRD4 (0.60) DRD2DRD4HTR2AHTR2CHTR2B
SCHEMBL6031812 0.81 DRD4 (1.00) DRD2DRD4SIGMAR1
SCHEMBL12668155 0.80 GAA (0.59) DRD2
SCHEMBL5542706 0.80 DRD4 (0.77) DRD2DRD4HTR2AHTR2CHTR2B
SCHEMBL12385909 0.80 DRD4 (0.77) DRD2DRD4LMNAHTR2AHTR2C
SCHEMBL10438222 0.78 DRD4 (0.64) DRD2DRD4HTR2AHTR2CHTR2B
SCHEMBL588149 0.78 DRD4 (1.00) DRD2DRD4LMNAHTR2CL3MBTL1
SCHEMBL6794331 0.78 DRD4 (0.79) DRD2DRD4HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012064569-A1 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-05-18 WO disclosed