SCHEMBL6442002

SCHEMBL6442002

NS(=O)(=O)c1ccc(N2CCN(Cc3ccccc3)CC2)cc1

nearest known ligand 0.66

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 3/20 0.66
CA1 P00915 13/20 0.64
CA2 P00918 13/20 0.64
CA9 Q16790 10/20 0.64
CA7 P43166 9/20 0.64
CA12 O43570 5/20 0.64
CA14 Q9ULX7 1/20 0.64
ALDH1A1 P00352 1/20 0.60
PTPN7 P35236 1/20 0.58
DUSP3 P51452 1/20 0.58
DRD2 P14416 1/20 0.58
HTR2A P28223 1/20 0.54
HTR2C P28335 1/20 0.54
HTR2B P41595 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4539301 0.85 DRD2 (0.73) DRD4DRD2HTR2AHTR2CHTR2B
SCHEMBL10438222 0.84 DRD4 (0.64) DRD4CA1CA2CA9CA12
SCHEMBL6031812 0.81 DRD4 (1.00) DRD4ALDH1A1DRD2
SCHEMBL26668277 0.80 CA1 (0.50) CA1CA2CA9CA7CA12
SCHEMBL5542706 0.80 DRD4 (0.77) DRD4DRD2HTR2AHTR2CHTR2B
SCHEMBL654308 0.80 DRD4 (0.77) DRD4DRD2HTR2AHTR2CHTR2B
Hydrochloric Acid SCHEMBL9742129 0.78 DRD4 (0.74) DRD4DRD2HTR2AHTR2CHTR2B
SCHEMBL588149 0.78 DRD4 (1.00) DRD4ALDH1A1DRD2HTR2C
SCHEMBL6794331 0.78 DRD4 (0.79) DRD4ALDH1A1DRD2HTR2AHTR2C
SCHEMBL19014647 0.78 BCL2 (0.64) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1226128-B1 NEW PYRIMIDINE-2,4,6-TRIONE DERIVATIVES, PROCESSES FOR THEIR PRODUCTION AND PHARMACEUTICAL AGENTS CONTAINING THESE COMPOUNDS HOFFMANN LA ROCHE (CH) 2005-02-23 EP disclosed
CN-1157382-C Novel pyrimidine-2, 4, 6-trione derivatives, process for their production and pharmaceutical agents containing these compounds - 2004-07-14 CN disclosed
US-6498252-B1 Pyrimidine-2,4,6-trione derivatives, processes for their production and pharmaceutical agents containing these compounds HOFFMANN-LA ROCHE INC. 2002-12-24 US disclosed
CN-1374954-A Novel pyrimidine-2, 4, 6-trione derivatives, process for their production and pharmaceutical agents containing these compounds HOFFMANN LA ROCHE (CH) 2002-10-16 CN disclosed
EP-1226128-A1 NEW PYRIMIDINE-2,4,6-TRIONE DERIVATIVES, PROCESSES FOR THEIR PRODUCTION AND PHARMACEUTICAL AGENTS CONTAINING THESE COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2002-07-31 EP disclosed
WO-2001025217-A1 NEW PYRIMIDINE-2,4,6-TRIONE DERIVATIVES, PROCESSES FOR THEIR PRODUCTION AND PHARMACEUTICAL AGENTS CONTAINING THESE COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2001-04-12 WO disclosed