SCHEMBL4539359

SCHEMBL4539359

CN(C)C1CCN(Cc2cc(C(N)(c3nc4cc(Oc5ccnc6[nH]ccc56)ccc4o3)N(C)C3CCN(Cc4cc(N)ccc4Cl)C3)ccc2Cl)C1

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDR P35968 14/20 0.52
BRAF P15056 3/20 0.34
EGFR P00533 2/20 0.34
MAPK14 Q16539 2/20 0.34
MAP3K7 O43318 1/20 0.34
MAP4K2 Q12851 1/20 0.34
CSK P41240 1/20 0.34
RAF1 P04049 1/20 0.33
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4539357 0.82 KDR (0.49) KDRBRAFEGFRMAPK14MAP3K7
SCHEMBL4364796 0.81 KDR (0.77) KDR
SCHEMBL4361243 0.68 KDR (1.00) KDR
SCHEMBL4371470 0.67 LTA4H (0.41)
SCHEMBL4364229 0.62 KDR (0.80) KDREGFR
SCHEMBL4365818 0.61 KDR (0.66) KDRBRAFRAF1
SCHEMBL4362982 0.61 KDR (1.00) KDR
SCHEMBL4361692 0.61 KDR (1.00) KDRMAP3K7
SCHEMBL4365782 0.60 KDR (0.84) KDR
SCHEMBL4375322 0.59 KDR (0.51) KDRBRAFMAPK14RAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7531553-B2 Heterocyclic compounds and methods of use AMGEN INC. (US) 2009-05-12 US disclosed