SCHEMBL4540378

SCHEMBL4540378

CC(=O)NC(C)c1ccc2c(c1)ncn2-c1cccc(-c2ccccc2C#N)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.61
GABRG2 P18507 1/20 0.61
GABRB3 P28472 1/20 0.61
GABRA5 P31644 1/20 0.61
GABRA3 P34903 1/20 0.61
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
PSEN1 P49768 1/20 0.41
PSEN2 P49810 1/20 0.41
APH1B Q8WW43 1/20 0.41
NCSTN Q92542 1/20 0.41
APH1A Q96BI3 1/20 0.41
PSENEN Q9NZ42 1/20 0.41
FGFR1 P11362 5/20 0.41
HPGD P15428 1/20 0.39
PPARG P37231 2/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
ALOX15 P16050 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1617241 1.00 GABRA1 (0.61) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL1616723 1.00 GABRA1 (0.61) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL1617363 0.90 GABRA1 (0.49) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL1616729 0.90 GABRA1 (0.49) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL1616031 0.87 NPC1 (0.46) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL1617011 0.87 NPC1 (0.46) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL1616776 0.86 NPC1 (0.53) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL1616093 0.86 NPC1 (0.53) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL1617120 0.86 NPC1 (0.53) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL1615890 0.85 ADRA2B (0.48) GABRA1GABRG2GABRB3GABRA5GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1996556-B1 BENZIMIDAZOLE DERIVATIVES AND THEIR USE FOR MODULATING THE GABAA RECEPTOR COMPLEX NEUROSEARCH AS (DK) 2009-11-18 EP claimed