SCHEMBL4540919

SCHEMBL4540919

O=C(CC1CCCN1C(=O)NCc1ccc(Cl)cc1Cl)NC12CCCC(CCC1)C2.[CH2]

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 8/20 0.46
P2RX7 Q99572 9/20 0.46
ALDH1A1 P00352 1/20 0.43
HRH3 Q9Y5N1 1/20 0.42
CYP2C9 P11712 1/20 0.41
CYP2J2 P51589 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4534910 0.88 EPHX2 (0.46) EPHX2P2RX7ALDH1A1HRH3CYP2C9
SCHEMBL8060069 0.84 EPHX2 (0.42) EPHX2P2RX7ALDH1A1HRH3CYP2C9
SCHEMBL8067140 0.80 EPHX2 (0.44) EPHX2P2RX7ALDH1A1HRH3CYP2C9
SCHEMBL4537295 0.79 ALDH1A1 (0.49) EPHX2P2RX7ALDH1A1HRH3CYP2C9
SCHEMBL4533493 0.76 ALDH1A1 (0.48) EPHX2P2RX7ALDH1A1HRH3CYP2C9
SCHEMBL8049790 0.75 EPHX2 (0.44) EPHX2P2RX7ALDH1A1HRH3
SCHEMBL4537463 0.75 EPHX2 (0.49) EPHX2P2RX7ALDH1A1HRH3CYP2C9
SCHEMBL4535274 0.74 EPHX2 (0.67) EPHX2ALDH1A1CYP2C9CYP2J2
SCHEMBL4542529 0.73 EPHX2 (0.59) EPHX2CYP2C9CYP2J2
SCHEMBL4537464 0.72 EPHX2 (0.51) EPHX2P2RX7ALDH1A1HRH3CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed