SCHEMBL4543449

SCHEMBL4543449

CC(C(N)=O)c1cn(C)c2ccc(O)cc12

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MTNR1B P49286 8/20 0.41
MTNR1A P48039 7/20 0.41
SPR P35270 1/20 0.41
IDO1 P14902 1/20 0.37
KDM4E B2RXH2 1/20 0.36
GAA P10253 2/20 0.35
PLA2G2A P14555 1/20 0.35
LMNA P02545 1/20 0.35
ICAM1 P05362 1/20 0.35
SELE P16581 1/20 0.35
WEE1 P30291 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2688129 0.87 KDM4E (0.43) MTNR1BMTNR1ASPRKDM4EGAA
SCHEMBL14502284 0.81 MTNR1B (0.43) MTNR1BMTNR1ASPRIDO1WEE1
SCHEMBL4092924 0.80 IDO1 (0.58) IDO1KDM4EGAALMNA
SCHEMBL31693354 0.75 KDM4E (0.45) MTNR1BMTNR1ASPRKDM4ELMNA
SCHEMBL18468650 0.74 MTNR1B (0.48) MTNR1BMTNR1ASPRGAALMNA
SCHEMBL5121452 0.73 SPR (0.50) MTNR1BMTNR1ASPRKDM4EPLA2G2A
SCHEMBL23809393 0.72 KDM4E (0.46) MTNR1BMTNR1AIDO1KDM4E
SCHEMBL7241953 0.71 KMT2A (0.48) KDM4E
SCHEMBL2007723 0.70 KMT2A (0.55) MTNR1BMTNR1ASPRGAALMNA
SCHEMBL23672305 0.70 MTNR1B (0.47) MTNR1BMTNR1ASPRGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2638034-A1 SUBSTITUTED HETEROAROMATIC CARBOXAMIDE AND UREA DERIVATIVES AS VANILLOID RECEPTOR LIGANDS Grünenthal GmbH (DE) 2013-09-18 EP disclosed
WO-2012062462-A1 SUBSTITUTED HETEROAROMATIC CARBOXAMIDE AND UREA DERIVATIVES AS VANILLOID RECEPTOR LIGANDS Grünenthal GmbH (DE) 2012-05-18 WO disclosed