SCHEMBL4545213

SCHEMBL4545213

O=C1C=C(c2ccc(O)cc2)Cc2cc(O)cc(O)c21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 8/20 0.41
ESR1 P03372 7/20 0.41
HSD17B1 P14061 3/20 0.37
GEMIN4 P57678 1/20 0.37
HSF1 Q00613 1/20 0.37
NPC1 O15118 1/20 0.37
MITF O75030 1/20 0.37
MAPT P10636 1/20 0.37
RAB9A P51151 1/20 0.37
ATM Q13315 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
BACE1 P56817 1/20 0.37
CA4 P22748 2/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA6 P23280 1/20 0.35
TDP2 O95551 1/20 0.35
CYP3A4 P08684 2/20 0.35
CYP19A1 P11511 2/20 0.35
MEN1 O00255 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13311725 0.88 APP (0.37) ESR2ESR1GEMIN4HSF1NPC1
SCHEMBL23571947 0.70 APP (0.37) MAPTBACE1CA4CA1CA2
SCHEMBL29586904 0.68 MAPT (0.47) ESR2ESR1GEMIN4HSF1NPC1
SCHEMBL22220312 0.67 BACE1 (0.68) ESR2ESR1NPC1MAPTBACE1
SCHEMBL5890294 0.67 NQO1 (0.62) ESR2ESR1NPC1MAPTRAB9A
SCHEMBL11921338 0.66 ESR1 (0.47) ESR2ESR1HSD17B1NPC1MAPT
SCHEMBL28032825 0.65 CES2 (0.49) ESR2ESR1TTR
SCHEMBL22789629 0.64 APP (0.37) ESR2ESR1MAPTNPSR1BACE1
SCHEMBL26346332 0.64 HSD17B1 (0.47) ESR2ESR1HSD17B1CA4CA1
SCHEMBL4179706 0.63 PBRM1 (0.44) ESR2HSD17B1MAPTCYP3A4TTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8716191-B2 Method of preparing an adduct UNIVERSITE DE STRASBOURG (FR) 2014-05-06 US disclosed
US-8716191-B2 Method of preparing an adduct UNIVERSITE DE STRASBOURG (FR) 2014-05-06 US disclosed
EP-2446033-B1 METHOD OF PREPARING AN ADDUCT UNIV STRASBOURG (FR) 2013-10-23 EP disclosed
US-20120115751-A1 METHOD OF PREPARING AN ADDUCT CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2012-05-10 US disclosed
US-20120115751-A1 METHOD OF PREPARING AN ADDUCT CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2012-05-10 US disclosed
WO-2010150103-A2 METHOD OF PREPARING AN ADDUCT UNIVERSITE DE STRASBOURG (FR) 2010-12-29 WO disclosed