SCHEMBL454624

SCHEMBL454624

O=POCO

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2975531 0.96
SCHEMBL9086436 0.74
SCHEMBL2403860 0.72
SCHEMBL5631310 0.67
SCHEMBL1109004 0.65 ALDH1A1 (0.33)
SCHEMBL3722742 0.65
Ammonia Solution, Strong SCHEMBL6702975 0.64
SCHEMBL454623 0.64
SCHEMBL2262997 0.62
SCHEMBL16533840 0.62

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 378 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2376507-B1 METHOD OF MAKING HYDROXYMETHYLPHOSPHONATES ICL IP AMERICA INC (US) 2013-05-15 EP claimed
EP-1554330-B1 PARTIALLY ESTER-EXCHANGED SIPM AND PROCESS THEREWITH INVISTA TECH SARL (CH) 2009-03-11 EP claimed
EP-1615934-B1 TITANIUM CHELATE DISPERSIONS DU PONT (US) 2007-06-27 EP claimed
US-7141559-B2 Glucocorticoid receptor ligands for the treatment of metabolic disorders KARO BIO AB (SE) 2006-11-28 US claimed
EP-1551860-B1 GLUCOCORTICOID RECEPTOR LIGANDS FOR THE TREATMENT OF METABOLIC DISORDERS KAROBIO AB (SE) 2006-11-22 EP claimed
EP-0184550-B1 5-AMINO-4-HYDROXY VALERYL AMIDE DERIVATIVES CIBA-GEIGY AG (CH) 1992-03-18 EP claimed
US-4727060-A HYPOTENSIVE AGENTS CIBA-GEIGY CORPORATION (US) 1988-02-23 US claimed
US-20240238774-A1 TWO COMPONENT ION EXCHANGE RESINS ION EXCHANGE (INDIA) LIMITED (IN) 2024-07-18 US disclosed
US-12012393-B2 Oxopiperazine derivatives Inthera Bioscience AG (CH) 2024-06-18 US disclosed
WO-2024119099-A1 GALLIUM-SALOPHEN ANTIMICROBIAL COMPOUNDS AND METHODS OF USE THEREOF UNIVERSITY OF MARYLAND, BALTIMORE (US) 2024-06-06 WO disclosed
EP-4373599-A1 TWO COMPONENT ION EXCHANGE RESINS Ion Exchange (India) Limited (IN) 2024-05-29 EP disclosed
EP-3544957-B1 DEGRADATION OF PROTEIN KINASES BY CONJUGATION OF PROTEIN KINASE INHIBITORS WITH E3 LIGASE LIGAND AND METHODS OF USE DANA FARBER CANCER INST INC (US) 2024-05-29 EP disclosed
US-20240158801-A1 STING DEPENDENT ADJUVANTS UNIVERSITY OF MIAMI 2024-05-16 US disclosed
CN-1165143-A Phosphosulfonate herbicides ROHM & HAAS (US) 1997-11-19 CN disclosed
US-5278193-A Ion exchange resin beads having aminoalkylphosphonic groups and processes for preparing them THE DOW CHEMICAL COMPANY (US) 1994-01-11 US disclosed
EP-0352949-B1 ION EXCHANGE RESIN BEADS AND PROCESSES FOR PREPARING THEM THE DOW CHEMICAL COMPANY (US) 1993-03-24 EP disclosed
EP-0184550-B1 5-AMINO-4-HYDROXY VALERYL AMIDE DERIVATIVES CIBA-GEIGY AG (CH) 1992-03-18 EP disclosed
US-4931591-A Novel 5-amino-4-hydroxyvaleryl derivatives CIBA-GEIGY CORPORATION (US) 1990-06-05 US disclosed
EP-0352949-A1 Ion exchange resin beads and processes for preparing them THE DOW CHEMICAL COMPANY (US) 1990-01-31 EP disclosed
US-4727060-A HYPOTENSIVE AGENTS CIBA-GEIGY CORPORATION (US) 1988-02-23 US disclosed