SCHEMBL4546719

SCHEMBL4546719

O=Nc1ccc(S(=O)(=O)Nc2cccc(-c3n[nH]cc3-c3ccncc3)c2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 2/20 0.47
PFKFB3 Q16875 2/20 0.43
ENPP1 P22413 1/20 0.42
AURKA O14965 8/20 0.42
AURKB Q96GD4 6/20 0.42
PDE4A P27815 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4C Q08493 1/20 0.41
PDE4D Q08499 1/20 0.41
NTRK1 P04629 1/20 0.41
MAP2K7 O14733 1/20 0.40
MAP2K4 P45985 1/20 0.40
PFKFB4 Q16877 1/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
HPGD P15428 1/20 0.40
HTT P42858 1/20 0.40
KMT2A Q03164 1/20 0.40
F2 P00734 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1850691 0.89 IMPDH2 (0.57) IMPDH2PFKFB3AURKAAURKBPDE4A
SCHEMBL1849634 0.88 CYP19A1 (0.52) IMPDH2PFKFB3ENPP1PDE4APDE4B
SCHEMBL1848921 0.88 ENPP1 (0.54) IMPDH2PFKFB3ENPP1AURKAAURKB
SCHEMBL13534569 0.88 HTR6 (0.50) IMPDH2PFKFB3ENPP1AURKAAURKB
SCHEMBL1847855 0.88 F2 (0.52) IMPDH2PFKFB3AURKAAURKBMAP2K7
SCHEMBL1847710 0.86 CYP19A1 (0.56) IMPDH2PFKFB3ENPP1AURKAAURKB
SCHEMBL1852646 0.86 ERAP1 (0.53) IMPDH2PFKFB3NTRK1MAP2K4MEN1
SCHEMBL1848169 0.85 SLC22A12 (0.47) IMPDH2PFKFB3ENPP1MAP2K4
SCHEMBL1849086 0.85 AURKA (0.51) IMPDH2PFKFB3AURKAAURKBMEN1
SCHEMBL1849348 0.84 CA12 (0.51) IMPDH2PFKFB3AURKAAURKBMAP2K7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2324008-B1 3,4-DIARYLPYRAZOLES AS PROTEIN KINASE INHIBITORS NERVIANO MEDICAL SCIENCES SRL (IT) 2012-05-09 EP disclosed