SCHEMBL4550512

SCHEMBL4550512

CC(NC(=O)c1ccnc(NC(=O)C2CC2)c1)c1cccc(O)c1

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BRAF P15056 2/20 0.55
GSK3B P49841 18/20 0.53
MAPT P10636 8/20 0.53
GSK3A P49840 9/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2715824 0.89 BRAF (0.55) BRAFGSK3BMAPTGSK3A
SCHEMBL18266733 0.87 ACACB (0.50)
SCHEMBL2715635 0.86 BRAF (0.59) BRAFGSK3BMAPTGSK3A
SCHEMBL2715632 0.86 BRAF (0.59) BRAFGSK3BMAPTGSK3A
SCHEMBL2714843 0.83 GSK3B (0.54) BRAFGSK3BMAPTGSK3A
SCHEMBL2715733 0.82 ROCK2 (0.49) BRAFGSK3BMAPTGSK3A
SCHEMBL2715734 0.82 ROCK2 (0.49) BRAFGSK3BMAPTGSK3A
SCHEMBL2713938 0.82 GSK3B (0.55) BRAFGSK3BMAPTGSK3A
SCHEMBL2717508 0.82 ROCK2 (0.49) BRAFGSK3BMAPTGSK3A
SCHEMBL18266201 0.80 ROCK2 (0.49) BRAFGSK3BMAPTGSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012053186-A1 ARYLAMIDE DERIVATIVES AS TTX-S BLOCKERS RAQUALIA PHARMA INC. (JP) 2012-04-26 WO disclosed