SCHEMBL4551325

SCHEMBL4551325

CCC(C#N)C1CN(C(=O)C(F)(F)F)CCc2cc(OC)ccc21

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.55
ESR2 Q92731 1/20 0.55
ABHD6 Q9BV23 1/20 0.46
MTNR1B P49286 5/20 0.41
CA1 P00915 3/20 0.41
CA2 P00918 3/20 0.41
CA9 Q16790 3/20 0.41
CA14 Q9ULX7 3/20 0.41
HSD11B1 P28845 1/20 0.41
DPP4 P27487 1/20 0.41
DPP8 Q6V1X1 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
DRD1 P21728 1/20 0.40
NOTUM Q6P988 1/20 0.39
GRIN2C Q14957 1/20 0.39
NQO2 P16083 3/20 0.38
MTNR1A P48039 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1094619 0.85 ESR1 (0.62) ESR1ESR2ABHD6MTNR1BCA1
SCHEMBL4551326 0.83 ESR1 (0.53) ESR1ESR2ABHD6MTNR1BHSD11B1
SCHEMBL1095554 0.82 ESR1 (0.61) ESR1ESR2ABHD6MTNR1BHSD11B1
SCHEMBL4937667 0.81 ESR1 (0.65) ESR1ESR2ABHD6MTNR1BCA1
SCHEMBL1095538 0.81 ESR1 (0.65) ESR1ESR2ABHD6MTNR1BCA1
SCHEMBL1095121 0.80 ESR1 (0.61) ESR1ESR2ABHD6MTNR1BCA1
SCHEMBL1095164 0.78 ESR1 (0.61) ESR1ESR2ABHD6MTNR1BHSD11B1
SCHEMBL6656989 0.77 ESR1 (0.60) ESR1ESR2ABHD6MTNR1BCA1
SCHEMBL2309023 0.74 ESR1 (0.85) ESR1ESR2ABHD6CA1CA2
SCHEMBL31164691 0.72 ESR1 (0.90) ESR1ESR2ABHD6CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2111859-A1 5HT2C receptor modulator compositions and methods of use Arena Pharmaceuticals, Inc. (US) 2009-10-28 EP disclosed