SCHEMBL4551326

SCHEMBL4551326

COc1ccc2c(c1)CCN(C(=O)C(F)(F)F)CC2CCCC#N

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.53
ESR2 Q92731 1/20 0.53
ABHD6 Q9BV23 1/20 0.44
MTNR1B P49286 2/20 0.41
NQO2 P16083 1/20 0.41
MTNR1A P48039 1/20 0.41
GRIN2B Q13224 1/20 0.41
SIGMAR1 Q99720 1/20 0.40
ABCB1 P08183 1/20 0.40
DPP4 P27487 1/20 0.40
DPP8 Q6V1X1 1/20 0.40
HSD11B1 P28845 1/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1095121 0.84 ESR1 (0.61) ESR1ESR2ABHD6MTNR1BNQO2
SCHEMBL1095554 0.84 ESR1 (0.61) ESR1ESR2ABHD6MTNR1BNQO2
SCHEMBL4551325 0.83 ESR1 (0.55) ESR1ESR2ABHD6MTNR1BNQO2
SCHEMBL1094619 0.81 ESR1 (0.62) ESR1ESR2ABHD6MTNR1BMTNR1A
SCHEMBL1095538 0.78 ESR1 (0.65) ESR1ESR2ABHD6MTNR1BHSD11B1
SCHEMBL4937667 0.78 ESR1 (0.65) ESR1ESR2ABHD6MTNR1BHSD11B1
SCHEMBL1095164 0.76 ESR1 (0.61) ESR1ESR2ABHD6MTNR1BNQO2
SCHEMBL6656989 0.75 ESR1 (0.60) ESR1ESR2ABHD6MTNR1BHSD11B1
SCHEMBL1094365 0.72 ESR1 (0.47) ESR1ESR2ABHD6MTNR1BNQO2
SCHEMBL2309023 0.72 ESR1 (0.85) ESR1ESR2ABHD6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2111859-A1 5HT2C receptor modulator compositions and methods of use Arena Pharmaceuticals, Inc. (US) 2009-10-28 EP disclosed