SCHEMBL4552450

SCHEMBL4552450

CCc1nn(Cc2ccc(OC)cc2)cc1Cl

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
KMT2A Q03164 1/20 0.45
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
ALOX15 P16050 1/20 0.42
CMA1 P23946 1/20 0.42
HSP90AA1 P07900 1/20 0.42
HSP90AB1 P08238 1/20 0.42
AADAT Q8N5Z0 1/20 0.42
NPBWR1 P48145 2/20 0.42
CYP19A1 P11511 2/20 0.41
DCTPP1 Q9H773 1/20 0.41
GSK3A P49840 1/20 0.41
GSK3B P49841 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
MCHR1 Q99705 1/20 0.40
PTGS2 P35354 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29339707 0.84 MEN1 (0.44) MEN1NPC1RAB9AKMT2AKDM4E
SCHEMBL19716279 0.81 MEN1 (0.47) MEN1NPC1RAB9AKMT2AKDM4E
SCHEMBL3359322 0.80 KMT2A (0.46) MEN1NPC1RAB9AKMT2ACMA1
SCHEMBL29339783 0.79 LTA4H (0.51) MEN1NPC1RAB9AKMT2AKDM4E
SCHEMBL370507 0.79 KMT2A (0.53) MEN1NPC1RAB9AKMT2ACMA1
SCHEMBL3357203 0.76 GSK3B (0.44) MEN1NPC1RAB9AKMT2ACMA1
SCHEMBL3356514 0.76 MAPT (0.46) MEN1KMT2AKDM4EALDH1A1MAPT
SCHEMBL29339883 0.75 AADAT (0.40) MEN1NPC1RAB9AKMT2AALDH1A1
SCHEMBL370625 0.75 MEN1 (0.44) MEN1NPC1RAB9AKMT2AKDM4E
SCHEMBL31052484 0.75 AADAT (0.49) MEN1NPC1RAB9AKMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2124943-A1 PYRAZOLO [3, 4-B]PYRIDINE DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS Ranbaxy Laboratories Limited (IN) 2009-12-02 EP disclosed
WO-2008111009-A1 PYRAZOLO [3, 4-B] PYRIDINE DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS RANBAXY LABORATORIES LIMITED (IN) 2008-09-18 WO disclosed