Camptothecin

Camptothecin

SCHEMBL4552875

CCCCCCl.CC[C@@]1(O)C(=O)OCc2c1cc1n(c2=O)Cc2cc3ccccc3nc2-1

nearest known ligand 0.85

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP1 P11387 18/20 0.85
ALDH1A1 P00352 4/20 0.85
MEN1 O00255 4/20 0.85
KMT2A Q03164 4/20 0.85
SMN1; SMN2 Q16637 4/20 0.85
KDM4E B2RXH2 3/20 0.85
GLA P06280 3/20 0.85
TP53 P04637 2/20 0.85
HPGD P15428 2/20 0.85
CYP3A4 P08684 2/20 0.85
HBB P68871 2/20 0.85
STAT6 P42226 1/20 0.85
CHEK1 O14757 1/20 0.85
HDAC3 O15379 1/20 0.85
ABCC4 O15439 1/20 0.85
GMNN O75496 1/20 0.85
LMNA P02545 1/20 0.85
CYP1A2 P05177 1/20 0.85
HNRNPA1 P09651 1/20 0.85
GAA P10253 1/20 0.85

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Camptothecin SCHEMBL6038 0.93 TOP1 (1.00) TOP1ALDH1A1MEN1KMT2ASMN1; SMN2
Camptothecin SCHEMBL28057307 0.93 TOP1 (1.00) TOP1ALDH1A1MEN1KMT2ASMN1; SMN2
Camptothecin SCHEMBL29360250 0.93 TOP1 (1.00) TOP1ALDH1A1MEN1KMT2ASMN1; SMN2
Camptothecin SCHEMBL788063 0.93 TOP1 (1.00) TOP1ALDH1A1MEN1KMT2ASMN1; SMN2
Camptothecin SCHEMBL4304557 0.93 TOP1 (1.00) TOP1ALDH1A1MEN1KMT2ASMN1; SMN2
Camptothecin SCHEMBL29369924 0.93 TOP1 (1.00) TOP1ALDH1A1MEN1KMT2ASMN1; SMN2
Camptothecin SCHEMBL2298909 0.93 TOP1 (1.00) TOP1ALDH1A1MEN1KMT2ASMN1; SMN2
Camptothecin SCHEMBL29351099 0.93 TOP1 (1.00) TOP1ALDH1A1MEN1KMT2ASMN1; SMN2
Camptothecin SCHEMBL3117386 0.92 TOP1 (0.98) TOP1ALDH1A1MEN1KMT2ASMN1; SMN2
Camptothecin SCHEMBL3651897 0.92 TOP1 (0.98) TOP1ALDH1A1MEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1435826-A4 DIAGNOSTIC OR THERAPEUTIC SOMATOSTATIN OR BOMBESIN ANALOG CONJUGATES AND USES THEREOF UNIV TULANE (US) 2009-07-15 EP disclosed
US-7326685-B2 Diagnostic or therapeutic somatostatin or bombesin analog conjugates and uses thereof THE ADMINISTRATORS OF THE TULANE EDUCATIONAL FUND (US) 2008-02-05 US disclosed
US-20050070470-A1 Diagnostic or therapeutic somatostatin or bombesin analog conjugates and uses thereof ADMINISTRATORS OF THE TULANE EDUCATIONAL FUND, THE 2005-03-31 US disclosed
EP-1435826-A2 DIAGNOSTIC OR THERAPEUTIC SOMATOSTATIN OR BOMBESIN ANALOG CONJUGATES AND USES THEREOF The Administrators of The Tulane Educational Fund (US) 2004-07-14 EP disclosed
WO-2003028527-A2 DIAGNOSTIC OR THERAPEUTIC SOMATOSTATIN OR BOMBESIN ANALOG CONJUGATES AND USES THEREOF THE ADMINISTRATORS OF THE TULANE EDUCATIONAL FUND (US) 2003-04-10 WO disclosed