SCHEMBL455312

SCHEMBL455312

CC(C)(C)c1ccc(NC(=S)NN=C2Nc3ccccc3C2=O)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.42
GAA P10253 3/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
TDP1 Q9NUW8 1/20 0.42
NPSR1 Q6W5P4 2/20 0.38
ALDH1A1 P00352 2/20 0.38
CFTR P13569 1/20 0.38
LMNA P02545 1/20 0.37
ALOX12 P18054 1/20 0.37
HTT P42858 1/20 0.37
XBP1 P17861 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NPC1 O15118 1/20 0.36
AKT1 P31749 1/20 0.36
TNKS O95271 1/20 0.36
TNKS2 Q9H2K2 1/20 0.36
PARP3 Q9Y6F1 1/20 0.36
CCKAR P32238 1/20 0.36
CCKBR P32239 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL456909 0.89 BCHE (0.43) MAPTGAAMEN1KMT2AALDH1A1
SCHEMBL2877739 0.87 MAPT (0.51) MAPTGAAMEN1KMT2ATDP1
SCHEMBL2877863 0.85 ALDH1A1 (0.46) MAPTGAAMEN1KMT2AALDH1A1
SCHEMBL456608 0.84 CYP1A2 (0.49) MAPTGAAMEN1KMT2ATDP1
SCHEMBL457421 0.84 LRRK2 (0.42) MAPTGAAMEN1KMT2ATDP1
SCHEMBL469876 0.84 KDR (0.46) MAPTGAAMEN1KMT2ATDP1
SCHEMBL455238 0.84 RAB9A (0.44) MAPTGAATDP1ALDH1A1CFTR
SCHEMBL455695 0.84 SLC2A1 (0.44) MAPTGAAMEN1KMT2ATDP1
SCHEMBL456579 0.83 ALDH1A1 (0.51) MAPTGAAMEN1KMT2ATDP1
SCHEMBL455700 0.81 ALDH1A1 (0.47) MAPTGAAMEN1KMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012033601-A1 THIOSEMICARBAZONES WITH MDR1 - INVERSE ACTIVITY THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH & HUMAN SERVICES (US) 2012-03-15 WO disclosed